Search Count: 13
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Rg7109 (N-{4-[6-Tert-Butyl-5-Methoxy-8-(6-Methoxy-2-Oxo-2,5-Dihydropyridin-3-Yl)Quinolin-3-Yl]Phenyl}Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-05-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 28L |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: ZN, 28L
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Compound 48 (N-({(3S)-1-[6-Tert-Butyl-5-Methoxy-8-(2-Oxo-1,2-Dihydropyridin-3-Yl)Quinolin-3-Yl]Pyrrolidin-3-Yl}Methyl)Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-05-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DMS, 28M |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: DMS, 28M
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The Crystal Structure Of Dyrk1A With A Bound Pyrido[2,3-D]Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2C3, 1PE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: 2C3, 1PE, SO4
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The Crystal Structure Of Dyrk1A With A Bound Pyrido[2,3-D]Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2C4, 1PE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: 2C4, 1PE, SO4
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Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(3,4,5-Trimethoxy-Phenyl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Isopropylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-10-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1B4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-30
Ligands: 1B4
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Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(6-Chloro-1-Methyl-1H-Indazol-3-Yl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Isopropylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2013-10-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1B5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-30
Ligands: 1B5
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Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(5,6,7,8-Tetrahydro-Imidazo[1,5-A]Pyridin-1-Yl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Tert-Butylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-10-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1B6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-30
Ligands: 1B6
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Crystal Structure Of Spleen Tyrosine Kinase Complexed With 6-((1R,2S)-2-Amino-Cyclohexylamino)-4-(6-Ethyl-Pyridin-2-Ylamino)-Pyridazine-3-Carboxylic Acid Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-07-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0VH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: 0VH
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Crystal Structure Of Jnk1Beta-Jip In Complex With An Azaquinolone Inhbitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2013-05-29 Classification: Transferase/Transferase Inhibitor Ligands: 0NR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 0NR
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-1,2,2-Trimethyl-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: PHU, 933 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: PHU, 933
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-2-Hydroxy-1,2-Dimethyl-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19Q
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((R)-2-Hydroxy-1,2-Dimethyl-Propyl
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19R
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((R)-1-Methyl-2-Oxo-2-Piperidin-1-Yl-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19S