Search Count: 15
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Crystal Structure Of The Bromodomain Of Atad2 With Az13824374
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 96L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 96L
 |
Crystal Structure Of The Bromodomain Of Atad2 With Phenol Hts Hit (Cpd 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 963 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 963
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Crystal Structure Of The Bromodomain Of Atad2 With Triazolopyridine (Cpd 14)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 95O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 95O
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Crystal Structure Of The Bromodomain Of Atad2 With Triazolopyridazine (Cpd 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 93L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 93L
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Bivalent Binding To Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2016-09-28 Classification: TRANSCRIPTION Ligands: ETU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: ETU
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Bivalent Binding To Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2016-09-28 Classification: TRANSCRIPTION Ligands: K6K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: K6K
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The First Bet Bromodomain Of Brd4 Bound To Compound 13 In A Bivalent Manner
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2016-09-21 Classification: Transcription Factor Ligands: XNH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: XNH, GOL
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 1.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: GQD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: GQD
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 2.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: QHG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: QHG
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: J0W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: J0W
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 4.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: 7QN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 7QN
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Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 5.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: VQI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: VQI
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A Novel Oral Selective Estrogen Receptor Down-Regulator, Azd9496, Drives Tumour Growth Inhibition In Estrogen Receptor Positive And Esr1 Mutant Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2015-12-16 Classification: SIGNALING PROTEIN Ligands: KE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: KE9
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: XBR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: XBR
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Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: GW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: GW5