Search Count: 18
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Plk1 Surface Entropy Reduction (Ser) Mutant In Complex With Inhibitor Bi 2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2025-11-26 Classification: TRANSFERASE Ligands: R78, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-26
Ligands: R78, SO4, GOL
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Crystal Structure Of Wild-Type Plk1 Kinase Domain In Complex With Thiazolidinone Inhibitor Compound 1 And A Selective Darpin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2025-11-26 Classification: TRANSFERASE Ligands: R78, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-26
Ligands: R78, GOL
 |
Crystal Structure Of The Second Bromodomain (Bd2) Of Human Brd2 Bound To Bi2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2021-11-17 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, R78, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: EDO, R78, CL
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Crystal Structure Of The Second Bromodomain (Bd2) Of Human Taf1 Bound To Plk1 Kinase Inhibitor Bi2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2021-09-22 Classification: GENE REGULATION Ligands: R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: R78
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Crystal Structure Of The First Bromodomain (Bd1) Of Human Brd2 Bound To Bi2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-08-11 Classification: GENE REGULATION Ligands: R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: R78
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Crystal Structure Of The Second Bromodomain (Bd2) Of Human Brd3 Bound To Bi2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-07-07 Classification: GENE REGULATION Ligands: R78, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: R78, EDO
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Crystal Structure Of Pi5P4Kiialpha Complex With Bi-2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-06-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R78, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: R78, SO4
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Crystal Structure Of Cgd4-650 With Compound Bi2536
Organism: Cryptosporidium parvum (strain iowa ii)
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2018-10-10 Classification: BIOSYNTHETIC PROTEIN Ligands: R78 |
Organism: Cryptosporidium parvum (strain iowa ii)
Method: X-RAY DIFFRACTION
Release Date: 2018-10-10
Ligands: R78
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Crystal Structure Of Cryptosporidium Parvum Bromodomain Cgd2_2690
Organism: Cryptosporidium parvum
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2018-04-18 Classification: TRANSFERASE Ligands: R78, GOL, UNX, SO4 |
Organism: Cryptosporidium parvum
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: R78, GOL, UNX, SO4
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Crystal Structure Of The First Bromodomain Of Human Brdt In Complex With Bi2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-04-04 Classification: TRANSCRIPTION/INHIBITOR Ligands: R78, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: R78, CL, EDO
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Crystal Structure Of The Human Camkk2B In Complex With Bi2526
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-12-13 Classification: TRANSFERASE Ligands: R78, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: R78, ACT
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First Bromodomain From Leishmania Donovani Ldbpk.091320 Complexed With Bi-2536
Organism: Leishmania donovani (strain bpk282a1)
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-10-05 Classification: UNKNOWN FUNCTION Ligands: R78, EDO |
Organism: Leishmania donovani (strain bpk282a1)
Method: X-RAY DIFFRACTION
Release Date: 2016-10-05
Ligands: R78, EDO
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Crystal Structure Analysis Of Pp-Brd20 From Tb427Tmp Complexed With Bi-2536
Organism: Trypanosoma brucei gambiense (strain mhom/ci/86/dal972)
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-07-22 Classification: GENE REGULATION Ligands: R78, UNX |
Organism: Trypanosoma brucei gambiense (strain mhom/ci/86/dal972)
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: R78, UNX
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Crystal Structure Of Bromodomain Of Pfa0510W From Plasmodium Falciparum
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-04-30 Classification: PROTEIN BINDING Ligands: R78, EDO |
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Release Date: 2014-04-30
Ligands: R78, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Bi 2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2014-03-05 Classification: TRANSCRIPTION/INHIBITOR Ligands: R78, EDO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-05
Ligands: R78, EDO, PEG
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Bi-2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-02-26 Classification: TRANSCRIPTION/INHIBITOR Ligands: EDO, R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-26
Ligands: EDO, R78
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: R78
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Structure Of Plk1 In Complex With Bi2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2008-02-05 Classification: TRANSFERASE Ligands: ZN, R78, TLA, SRT, TAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-05
Ligands: ZN, R78, TLA, SRT, TAR