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7OE8 image
C-Terminal Bromodomain Of Human Brd2 With N5-((1R,5S,6R)-3-Oxabicyclo[3.1.0]Hexan-6-Yl)-3-(1H-Indol-4-Yl)-N7-Methyl-2,3-Dihydrobenzofuran-5,7-Dicarboxamide

7OE9 image
C-Terminal Bromodomain Of Human Brd2 With Rac-N5-((1R,5S)-3-Oxabicyclo[3.1.0]Hexan-6-Yl)-N7,3-Dimethyl-3-Phenyl-2,3-Dihydrobenzofuran-5,7-Dicarboxamide

6SWN image
N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd1 (Gsk778)

6SWO image
C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd1 (Gsk778)

6SWP image
C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd2 (Gsk046)

6SWQ image
N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd2 (Gsk046)

5FP7 image
Crystal Structure Of Human Kdm4D In Complex With 3-4-Methylthiophen-2- Yl Methylaminopyridine-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2016-11-09
Classification: INHIBITOR
Ligands: ZN, FE2, GOL, YC8, SO4

5LMA image
Human Spleen Tyrosine Kinase Kinase Domain In Complex With Azanaphthyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.43 Å Release Date: 2016-09-14
Classification: TRANSFERASE
Ligands: 6ZG, GOL, DMS

5LMB image
Human Spleen Tyrosine Kinase Kinase Domain In Complex With Azanaphthyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2016-09-14
Classification: TRANSFERASE
Ligands: 6ZF, GOL

5FP3 image
Cell Penetrant Inhibitors Of The Jmjd2 (Kdm4) And Jarid1 (Kdm5) Families Of Histone Lysine Demethylases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2016-01-27
Classification: OXIDOREDUCTASE
Ligands: YC8, ZN, MG, BCN, CO

5FP4 image
Crystal Structure Of Human Kdm4D In Complex With 3-(4- Phenylbutanamido)Pyridine-4-Carboxylic Acid

5FP8 image
Crystal Structure Of Human Kdm4D In Complex With 3-4-Methylthiophen-2- Ylmethylaminopyridine-4-Carboxylic Acid

5FP9 image
Crystal Structure Of Human Kdm4D In Complex With 3-Aminopyridine-4- Carboxylic Acid

5FPA image
Crystal Structure Of Human Kdm4D In Complex With 3H,4H-Pyrido-3,4-D- Pyrimidin-4-One

5FPB image
Crystal Structure Of Human Kdm4D In Complex With 2-1H-Pyrazol-4-Yloxy- 3H,4H-Pyrido-3,4-D-Pyrimidin-4-One

4YJO image
The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000222
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: 4DF, GOL

4YJP image
The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000223
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: 4DL, DMS

4YJQ image
Syk Kinase Domain In Complex With Inhibitor Gtc000224
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.34 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: 4DK

4YJR image
Syk Kinase Domain In Complex With Inhibitor Gtc000225
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.32 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: 4DJ

4YJS image
The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000226
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.22 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: 4DN
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