Search Count: 67
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G-925 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2022-08-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GGU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: GGU
 |
G-059 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2022-08-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GJN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: GJN
 |
Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.13 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: QRY, CL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: QRY, CL, SO4
 |
Crystal Structure Of The P300 Acetyltransferase Domain With Peptide-Competitive Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA, QS4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: COA, QS4, DMS
 |
Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: SO4, CL, QS1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: SO4, CL, QS1
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Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: QSD, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: QSD, SO4, CL
 |
Crystal Structure Of The P300 Acetyltransferase Domain With Allosteric Inhibitor Cpi-090 And Coa
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2019-10-23 Classification: TRANSFERASE/INHIBITOR Ligands: COA, OJ7 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: COA, OJ7
 |
Crystal Structure Of The P300 Acetyltransferase Domain With Allosteric Inhibitor Cpi-076 And Coa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-10-23 Classification: TRANSFERASE/INHIBITOR Ligands: COA, OK7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: COA, OK7
 |
Taf1-Bd2 In Complex With Cpd27 (6-(But-3-En-1-Yl)-4-(1-Methyl-6-(Morpholine-4-Carbonyl)-1H-Benzo[D]Imidazol-4-Yl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-11-14 Classification: Transcription/Inhibitor Ligands: G9V |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: G9V
 |
Taf1-Bd2 In Complex With Cpd8 (6-(But-3-En-1-Yl)-4-(3-(Morpholine-4-Carbonyl)Phenyl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-31 Classification: Transcription/Inhibitor Ligands: G9Y |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: G9Y
 |
Crystal Structure Of The Bromodomain Of Human Crebbp Bound To Pyrazolopiperidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XB, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XB, DMS
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Crebbp Bromodomain In Complex With Cpd 44 (3-((5-Acetyl-1-(Cyclopropylmethyl)-4,5,6,7-Tetrahydro-1H-Pyrazolo[4,3-C]Pyridin-3-Yl)Amino)-N-Isopropylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.09 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XG, EDO
 |
Crebbp Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XH, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XH, EDO, DMS
 |
Brd4 Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: EDO, DMS, GOL, PEG, 6XH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: EDO, DMS, GOL, PEG, 6XH
 |
Brd9 In Complex With Cpd1 (6-Methyl-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2016-10-12 Classification: RNA BINDING PROTEIN Ligands: EDO, PEG, 67N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: EDO, PEG, 67N
 |
Brd9 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2016-10-12 Classification: RNA BINDING PROTEIN Ligands: 67B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 67B
 |
Brd9 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 69G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 69G
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Brd4 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 67B, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 67B, EDO, DMS
 |
Brd4 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: PGE, EDO, DMS, 69G, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: PGE, EDO, DMS, 69G, GOL
 |
Structure Of G9A Set-Domain With Histone H3K9Norleucine Mutant Peptide And Bound S-Adenosylmethionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2016-09-14 Classification: TRANSFERASE Ligands: ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: ZN, SAM