Search Count: 35
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Crystal Structure Of 6-Fluoropyrazolo[1,5-A]Pyridine Derivative Bound To Kit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1DJF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1DJF
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Crystal Structure Of Casdatifan Bound To Hif2A-B*:Arnt-B* Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2026-02-18 Classification: TRANSCRIPTION Ligands: A1I0H, FMT, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: A1I0H, FMT, MG
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Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2021-11-03 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V84 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: V84
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With The Ampcp Derivative A894 (Compound 2N In Publication) In The Closed Form (Crystal Form Iv)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2021-01-20 Classification: HYDROLASE Ligands: ZN, OO2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: ZN, OO2
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With The Ampcp Derivative A1202 (Compound 4A In Publication) In The Closed Form (Crystal Form Iv)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-01-20 Classification: HYDROLASE Ligands: ZN, OO5, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: ZN, OO5, CA
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Crystal Structure Of Human Pi3K-Gamma In Complex With Inhibitor Ipi-549
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V7Y, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V7Y, SO4
 |
Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V81, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V81, SO4
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative Ab680 (Compound 55 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-09-16 Classification: HYDROLASE Ligands: ZN, CA, QDH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: ZN, CA, QDH
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative A830 (Compound 16 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-07-22 Classification: HYDROLASE Ligands: ZN, CA, QCQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ZN, CA, QCQ
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2396 (Compound 74 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1H
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2410 (Compound 53 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1Q
 |
Human Ecto-5'-Nucleotidase (Cd73) In Complex With A1618 (Compound 1B In Publication) In The Closed State In Crystal Form Iii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, O1T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, O1T
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Co-Crystal Structure Of Mdm2 With Inhibitor (2S,5R,6S)-2-Benzyl-5,6-Bis(4-Bromophenyl)-4-Methylmorpholin-3-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-05-01 Classification: LIGASE/LIGASE INHIBITOR Ligands: 1MN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 1MN, SO4
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Co-Crystal Structure Of Mdm2 With Inhibitor (2S,5R,6S)-2-Benzyl-5,6-Bis(4-Chlorophenyl)-4-Methylmorpholin-3-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-05-01 Classification: LIGASE/LIGASE INHIBITOR Ligands: 1MO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 1MO, SO4
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Co-Crystal Structure Of Mdm2 With Inhibitor (2R,3E)-2-[(2S,3R,6S)-2,3-Bis(4-Chlorophenyl)-6-(4-Fluorobenzyl)-5-Oxomorpholin-4-Yl]Pent-3-Enoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-05-01 Classification: LIGASE/LIGASE INHIBITOR Ligands: 1MQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 1MQ
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Co-Crystal Structure Of Mdm2 With Inhibitor (2'S,3R,4'S,5'R)-N-(2-Aminoethyl)-6-Chloro-4'-(3-Chloro-2-Fluorophenyl)-2'-(2,2-Dimethylpropyl)-2-Oxo-1,2-Dihydrospiro[Indole-3,3'-Pyrrolidine]-5'-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-05-01 Classification: LIGASE/LIGASE INHIBITOR Ligands: 1MT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 1MT
 |
Co-Crystal Structure Of Mdm2 With Inhibitor {(2S,5R,6S)-6-(3-Chlorophenyl)-5-(4-Chlorophenyl)-4-[(2S)-1-Hydroxybutan-2-Yl]-3-Oxomorpholin-2-Yl}Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-05-01 Classification: LIGASE/LIGASE INHIBITOR Ligands: 1MY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 1MY
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase 1 (11B-Hsd1) In Complex With 4,4-Disubstituted Cyclohexylbenzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-10-05 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: 3PJ, NAP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: 3PJ, NAP
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Crystal Structure Of 11Beta-Hydroxysteroid Dehydrogenase-1 (11B-Hsd1) In Complex With Diarylsulfone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-07-20 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 3OQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-07-20
Ligands: NAP, 3OQ
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Crystal Structure Of 11Beta-Hydroxysteroid Dehydrogenase 1 (11B-Hsd1) In Complex With Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2009-12-01 Classification: OXIDOREDUCTASE Ligands: NAP, IIG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-01
Ligands: NAP, IIG