Search Count: 21
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
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Co-Crystal Structure Of Perk Bound To N-{5-[(6,7-Dimethoxyquinolin-4-Yl)Oxy]Pyridin-2-Yl}-1-Methyl-3-Oxo-2-Phenyl-5-(Pyridin-4-Yl)-2,3-Dihydro-1H-Pyrazole-4-Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z2, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 3Z2, SO4
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Co-Crystal Structure Of Perk With 2-Amino-N-[4-Methoxy-3-(Trifluoromethyl)Phenyl]-4-Methyl-3-[2-(Methylamino)Quinazolin-6-Yl]Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-01-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z1, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: 3Z1, TLA
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Co-Crystal Structure Of Perk Bound To 4-{2-Amino-3-[5-Fluoro-2-(Methylamino)Quinazolin-6-Yl]-4-Methylbenzoyl}-1-Methyl-2,5-Diphenyl-1,2-Dihydro-3H-Pyrazol-3-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-01-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z3, TLA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: 3Z3, TLA, GOL
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Co-Crystal Structure Of Perk Bound To 4-{2-Amino-4-Methyl-3-[2-(Methylamino)-1,3-Benzothiazol-6-Yl]Benzoyl}-1-Methyl-2,5-Diphenyl-1,2-Dihydro-3H-Pyrazol-3-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-01-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z4, TLA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: 3Z4, TLA, GOL
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Co-Crystal Structure Of Perk Bound To 4-[2-Amino-4-Methyl-3-(2-Methylquinolin-6-Yl)Benzoyl]-1-Methyl-2,5-Diphenyl-1,2-Dihydro-3H-Pyrazol-3-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-01-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z5, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: 3Z5, TLA
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Co-Crystal Structure Of Perk Bound To 1-[5-(4-Amino-2,7-Dimethyl-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl)-2,3-Dihydro-1H-Indol-1-Yl]-2-[3-Fluoro-5-(Trifluoromethyl)Phenyl]Ethanone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-01-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: 3Z6
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Nmr Solution Structure Of Pin1 Ww Domain Mutant 5-1
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2013-06-26
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Nmr Solution Structure Of Pin1 Ww Domain Mutant 5-1G
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2013-06-26 Classification: ISOMERASE Ligands: NAG |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2013-06-26
Ligands: NAG
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Nmr Solution Structure Of Pin1 Ww Domain Variant 6-1
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2013-06-26
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Nmr Solution Structure Of Pin1 Ww Domain Mutant 6-1G
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2013-06-26 Classification: ISOMERASE Ligands: NAG |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2013-06-26
Ligands: NAG
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X-Ray Co-Crystal Structure Of 2-Amino-6-Phenylpyrimido[5',4':5,6]Pyrimido[1,2-A]Benzimidazol-5(6H)-One 25 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-12-30 Classification: TRANSFERASE Ligands: SO4, AM9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-30
Ligands: SO4, AM9
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X-Ray Co-Crystal Structure Aminobenzimidazole Triazine 1 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-09-16 Classification: TRANSFERASE Ligands: SO4, AM0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-09-16
Ligands: SO4, AM0
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Co-Crystal Structure Of Lck And Aminopyrimidine Amide 10B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-09-16 Classification: TRANSFERASE Ligands: AM5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-09-16
Ligands: AM5
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Co-Crystal Structure Of Lck And Aminopyrimidine Reverse Amide 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-09-16 Classification: TRANSFERASE Ligands: AM6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-09-16
Ligands: AM6
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X-Ray Crystal Structure Of 2-Aminopyrimidine Carbamate 43 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-02-27 Classification: TRANSFERASE Ligands: SO4, 1N9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: SO4, 1N9
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Crystal Structure Of Aminoquinazoline 1 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-02-27 Classification: TRANSFERASE Ligands: 242 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: 242
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Crystal Structure Of Aminoquinazoline 36 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-02-27 Classification: TRANSFERASE Ligands: 1N8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: 1N8
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Crystal Structure Of P38 Alpha In Complex With A Selective Pyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-04-26 Classification: TRANSFERASE Ligands: SO4, 6NP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-04-26
Ligands: SO4, 6NP