Search Count: 29
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Crystal Structure Of Human Tlr8 Ectodomain Bound To Small Molecule Antagonist 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2022-05-04 Classification: RNA BINDING PROTEIN Ligands: NAG, RQY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: NAG, RQY
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Crystal Structure Of The Human Brd2 Bd1 Bromodomain In Complex With 9-(Cyclopropylmethyl)-7-[(2R,6S)-2,6-Dimethylmorpholine-4-Carbonyl]-3-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-9H-Carbazole-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW1, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 9-Benzyl-2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW4, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW7, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW7, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Bms-986158, 2-{3-(1,4-Dimethyl-1H-1,2,3-Triazol-5-Yl)-5-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-5H-Pyrido[3,2-B]Indol-7-Yl}Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YWA, IOD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YWA, IOD, EDO
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Crystal Structure Of Human Tlr8 Ectodomain Bound To Small Molecule Antagonist 14C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2020-08-12 Classification: RNA BINDING PROTEIN Ligands: NAG, QSM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: NAG, QSM
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Crystal Structure Of Irak-4 With A 4,6-Diaminonicotinamide Inhibitor (Compound Number 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-10-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9YY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: 9YY
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Crystal Structure Of Irak-4 With A 4,6-Diaminonicotinamide Inhibitor (Compound Number 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-10-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9YS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: 9YS
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Crystal Structure Of Jak3 Kinase Domain With A 4,6-Diaminonicotinamide Inhibitor (Compound Number 7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2017-10-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9YV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: 9YV
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Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 9EM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 9EM
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Crystal Structure Of Pi3K Alpha In Complex With A 7-(3-(Piperazin-1-Yl)Phenyl)Pyrrolo[2,1-F][1,2,4] Triazin-4-Amine Deriviatine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-02-08 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 85S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: 85S
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Crystal Structure Of Pi3K Delta In Complex With A 7-(3-(Piperazin-1-Yl)Phenyl)Pyrrolo[2,1-F][1,2,4] Triazin-4-Amine Deriviatine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2017-02-08 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 85S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: 85S
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Crystal Structure Of Cyclin-Dependent Kinase 2 (Cdk2-Wt) Complex With (2S)-N-(5-(((5-Tert-Butyl-1,3-Oxazol-2-Yl)Methyl)Sulfanyl)-1,3-Thiazol-2-Yl)-2-Phenylpropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-10-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1YG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: 1YG
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The Crystal Structure Of Apo Human Hdhd4 From Se-Mad
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2013-06-26 Classification: HYDROLASE Ligands: PO4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: PO4, MG
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The Crystal Structure Of Human Hdhd4 In Complex With Magnesium And The Phosphate Mimetic Vanadate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-06-26 Classification: HYDROLASE Ligands: VO4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: VO4, MG
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With N-(N-(4-Amino-3,5- Dichlorobenzyl)Carbamimidoyl)-3-(4-Methoxyphenyl)-5- Methyl-4-Isothiazolecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-10-10 Classification: HYDROLASE/INHIBITOR Ligands: 0VA, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0VA, IOD
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Db-Mut) Complex With N-(N-(4- Acetamido-3-Chloro-5-Methylbenzyl)Carbamimidoyl)-3-(4- Methoxyphenyl)-5-Methyl-4-Isothiazolecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-10-10 Classification: HYDROLASE/INHIBITOR Ligands: 0VB, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0VB, IOD
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Crystal Structure Of Influenza A Virus Nucleoprotein With Ligand
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2012-08-29 Classification: VIRAL PROTEIN/INHIBITOR Ligands: 0MM |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 0MM
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Crystal Structure Of Influenza A Virus Nucleoprotein With Ligand
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2011-09-14 Classification: VIRAL PROTEIN Ligands: LGH |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 2011-09-14
Ligands: LGH
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Crystal Structure Of The Hepatitis C Virus Ns5B Rna-Dependent Rna Polymerase Complex With (2E)-3-(4-{[(1-{[(13-Cyclohexyl-6-Oxo-6,7-Dihydro-5H-Indolo[1,2-D][1,4]Benzodiazepin-10-Yl)Carbonyl]Amino}Cyclopentyl)Carbonyl]Amino}Phenyl)Prop-2-Enoic Acid
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2011-04-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 23E, SO4 |
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: 23E, SO4