Search Count: 57
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-(Difluorom Ethoxy)-4-(1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YFV, SO4, 5OI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: YFV, SO4, 5OI
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand 2-(1-Amino-3-Methylbutyl)-6- (Pyridin-4-Yl)Quinoline-4-Carbonitrile
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5P6, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: 5P6, SO4
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-(Difluorom Ethoxy)-4-(1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5QI, PG6, SO4, YFV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: 5QI, PG6, SO4, YFV
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Crystal Structure Of Mripk3 Complexed With N-(3-Fluoro-4-{1H-Pyrrolo[2,3-B]Pyridin-4-Yloxy}Phenyl)-1-(4-Fluorophenyl)-2-Oxo-1,2-Dihydropyridine-3-Carboxamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: 1FN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: 1FN
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Btk In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2019-04-03 Classification: TRANSFERASE/INHIBITOR Ligands: LTJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: LTJ
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Crystal Structure Of Gsk3B In Complex With Compound 15: 2-[(Cyclopropylcarbonyl)Amino]-N-(4-Methoxypyridin-3-Yl)Pyridine-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 3UO
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Crystal Structure Of Gsk3B In Complex With Compound 18: 2-[(Cyclopropylcarbonyl)Amino]-N-(4-Phenylpyridin-3-Yl)Pyridine-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 3UP
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Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With Bms-824171 Aka 6-[(3R)-3-(4-Tert-Bu Tylbenzamido)Piperidin-1-Yl]-2-{[4-(Morpholine-4-Carbonyl) Phenyl]Amino}Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2015-09-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4UQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 4UQ
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Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With Bms-824171 Aka 6-[(3R)-3-(4-Tert-Bu Tylbenzamido)Piperidin-1-Yl]-2-{[4-(Morpholine-4-Carbonyl) Phenyl]Amino}Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2015-09-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4US, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 4US, DMS, EDO
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Crystal Structure Of Xiap-Bir2 Domain Complexed With (S)-3-(4-Methoxyphenyl)-2-((S)-2-((S)-1-((S)-2-((S)-2-(Methylamino)Propanamido)Pent-4-Ynoyl)Pyrrolidine-2-Carboxamido)-3-Phenylpropanamido)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2015-05-06 Classification: APOPTOSIS Ligands: ZN, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: ZN, SO4, GOL
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Structure Of A Carboxamide Compound (3) (2-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}-4-Oxo-4H-1Lambda~4~,3-Thiazole-5-Carboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WE
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Structure Of A Carvoxamide Compound (15) (N-[4-(Isoquinolin-7-Yl)Pyridin-2-Yl]Cyclopropanecarboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WF
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Structure Of A Carboxamine Compound (26) (2-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}-4-Methoxypyrimidine-5-Carboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WG
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Crystal Structure Of Xiap-Bir2 Domain Complexed With Ligand Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2015-03-04 Classification: APOPTOSIS Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-04
Ligands: ZN
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Crystal Structure Of Xiap-Bir2 Domain Complexed With Ligand Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2015-03-04 Classification: APOPTOSIS Ligands: ZN, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-04
Ligands: ZN, SO4, GOL
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Human Fdps Synthase In Complex With A Rigid Analog Of Risedronate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2011-06-29 Classification: TRANSFERASE Ligands: UNV, MG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-29
Ligands: UNV, MG, SO4
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Human Fdps Synthase In Complex With A N-Methyl Pyridinum Bisphosphonate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-06-01 Classification: TRANSFERASE Ligands: UNR, MG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-01
Ligands: UNR, MG, SO4
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 279 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 279
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 287 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 287
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Human Fdps Synthase In Complex With Minodronate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-11-06 Classification: TRANSFERASE Ligands: M0N, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: M0N, MG