Search Count: 26
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Crystal Structure Of Kat6A In Complex With Inhibitor Ctx-648 (Pf-9363)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2023-07-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R7L, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: R7L, ZN
 |
Optimization Of Tead P-Site Binding Fragment Hit Into In Vivo Active Lead Msc-4106
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JJU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JJU, SO4
 |
Human Tead3 In Complex With 1-Cyclopentyl-1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JIK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JIK
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Hbo1 Is Required For The Maintenance Of Leukaemia Stem Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-12-25 Classification: antitumor protein/inhibitor Ligands: ZN, GOL, JAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: ZN, GOL, JAV
 |
Hbo1 Is Required For The Maintenance Of Leukaemia Stem Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2019-12-25 Classification: antitumor protein/transferase Ligands: ZN, ACO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: ZN, ACO
 |
Wdr5Delta23 Bound To (2-Butyl-1H-Imidazol-4-Yl)Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: OHJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OHJ
 |
Wdr5Delta32 Bound To (2-Methyl-1H-Imidazol-4-Yl)Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: OHG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OHG, SO4
 |
Wdr5Delta32 Bound To Benzyl (4-(5-(Hydroxymethyl)-1H-Imidazol-2-Yl)Butyl)Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: OHV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OHV, SO4
 |
Wdr5Delta23 Bound To N-(4-(5-(Hydroxymethyl)-1H-Imidazol-2-Yl)Butyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: SO4, OH7, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: SO4, OH7, CL
 |
Wdr5Delta32 Bound To (2-(3-Methoxy-3-Phenylpropyl)-1H-Imidazol-4-Yl)Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: OH4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OH4, PEG
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Wdr5Delta23 Bound To (2-(3-Phenylpropyl)-1H-Imidazol-4-Yl)Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: OGY, CL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OGY, CL, SO4
 |
Wdr5Delta23 Bound To N-(4-(5-(Hydroxymethyl)-1H-Imidazol-2-Yl)Butyl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: OH1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OH1
 |
Wdr5Delta32 Bound To Methyl (4-(4-(Hydroxymethyl)-1H-Imidazol-2-Yl)Butyl)Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/Inhibitor Ligands: OGM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OGM, SO4
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Wdr5Delta32 Bound To N-(4-(5-(Hydroxymethyl)-1H-Imidazol-2-Yl)Butyl)-2-Phenylacetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/INHIBITOR Ligands: OJG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OJG, SO4
 |
Wdr5Delta32 Bound To Methyl Benzyl(4-(4-(Hydroxymethyl)-1H-Imidazol-2-Yl)Butyl)Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/INHIBITOR Ligands: SO4, OJJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: SO4, OJJ
 |
Wdr5Delta32 Bound To Peptidomimetic
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/INHIBITOR Ligands: OK4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OK4, SO4
 |
Wdr5Delta32 Bound To Ethyl 3-(4-(Hydroxymethyl)-1H-Imidazol-2-Yl)Propanoate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/INHIBITOR Ligands: OJM, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OJM, SO4, EDO
 |
Wdr5Delta32 Bound To N-(4-(4-(Hydroxymethyl)-1H-Imidazol-2-Yl)Butyl)Acrylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2019-12-11 Classification: PROTEIN BINDING/INHIBITOR Ligands: OJP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: OJP, SO4
 |
Design And Optimization Of Biaryl Ether Aryl Sulfonamides As Selective Inhibitors Of Nav1.7: Discovery Of Clinical Candidate Pf-05089771
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-06-07 Classification: OXIDOREDUCTASE Ligands: HEM, 6RJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: HEM, 6RJ
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Crystal Structure Of Trka In Complex With Pf-00593174
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-03-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 6K0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 6K0