Search Count: 11
![]() |
Pde10A With Imidazopyrazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-08-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, 6RC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: ZN, MG, 6RC
![]() |
Cfms Tyrosine Kinase In Complex With 4-Cyano-1H-Imidazole-2-Carboxylic Acid (2-Cyclohex-1-Enyl-4-Piperidin-4-Yl-Phenyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-12-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ACT, KRJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: ACT, KRJ
![]() |
Cfms Tyrosine Kinase In Complex With 5-Cyano-Furan-2-Carboxylic Acid [4-(4-Methyl-Piperazin-1-Yl)-2-Piperidin-1-Yl-Phenyl]-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-12-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KRL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: KRL, SO4
![]() |
Cyanofluorophenylacetamides As Orally Efficacious Thrombin Inhibitors
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2009-02-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DKK |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: DKK
![]() |
Cfms Tyrosine Kinase In Complex With A Pyridopyrimidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-02-17 Classification: TRANSFERASE Ligands: SO4, 8C5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: SO4, 8C5
![]() |
2-(2-Chloro-6-Fluorophenyl)Acetamides As Potent Thrombin Inhibitors
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-08-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: I50 |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2008-08-26
Ligands: I50
![]() |
Cfms Tyrosine Kinase (Tie2 Kid) In Complex With A Pyrimidinopyridone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2008-07-15 Classification: TRANSFERASE Ligands: SO4, IXH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-15
Ligands: SO4, IXH
![]() |
X-Ray Structure Of Fxa In Complex With 7-Fluoroindazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-01-29 Classification: HYDROLASE Ligands: JNJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: JNJ
![]() |
C-Fms Tyrosine Kinase In Complex With A Quinolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2006-11-28 Classification: TRANSFERASE Ligands: SO4, 6C3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: SO4, 6C3
![]() |
Cfms Tyrosine Kinase (Fgf Kid) In Complex With An Arylamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-11-28 Classification: TRANSFERASE Ligands: 5CN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: 5CN
![]() |
Cfms Tyrosine Kinase (Tie2 Kid) In Complex With An Arylamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2006-11-28 Classification: TRANSFERASE Ligands: 5CN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: 5CN
