Search Count: 31
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase In Complex With Amppnp And Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: A1AU3, GOL, MG, ANP, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: A1AU3, GOL, MG, ANP, ZN
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase In Complex With Amppnp And Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: MG, ZN, ANP, GOL, JUJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: MG, ZN, ANP, GOL, JUJ
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 5; 3-((2-((3-Chloro-4-Fluorophenyl)Amino)-2-Oxoethyl)Carbamoyl)Picolinic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ANP, A1BJH, ZN, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ANP, A1BJH, ZN, MN
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 36; (S)-(6,7-Dichloro-1-Methyl-1,3,4,5-Tetrahydro-2H-Pyrido[4,3-B]Indol-2-Yl)(5-(2-Hydroxyethoxy)Pyrimidin-2-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ZN, A1BJA, ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ZN, A1BJA, ANP, MN
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 23; (S)-1-(6,7-Dichloro-1-Methyl-1,3,4,5-Tetrahydro-2H-Pyrido[4,3-B]Indol-2-Yl)-2-Methoxyethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ZN, A1BJD, ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ZN, A1BJD, ANP, MN
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-07-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, PQI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: MG, GDP, PQI
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-07-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, PUO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: MG, GDP, PUO
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 51A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 51A
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 52R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 52R
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: MG, L9W, 54N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: MG, L9W, 54N
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Crystal Structure Of Cdk9-Cyclin T1 Bound By Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-10-27 Classification: TRANSFERASE Ligands: UT5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-27
Ligands: UT5
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Eed In Complex With A Cyano-Benzofuran
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: CA, L9W, PV5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: CA, L9W, PV5
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Eed In Complex With A Triazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: L9W, GOL, EJR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: L9W, GOL, EJR
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Cdk9-Cyclin-T1 Complex Bound By Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.37 Å Release Date: 2020-12-23 Classification: TRANSFERASE Ligands: Q6E, TRS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: Q6E, TRS, PO4
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Pi3Kg In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2019-01-30 Classification: TRANSFERASE Ligands: DD8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-30
Ligands: DD8
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Crystal Structure Of Myeloperoxidase Subform C (Mpo) Complex With Compound-6 Aka 7-(Benzyloxy)-1H-[1,2, 3]Triazolo[4,5-D]Pyrimidin-5-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-04-18 Classification: METAL BINDING PROTEIN Ligands: AEY, CL, HEM, CA, NAG, FUC, MAN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: AEY, CL, HEM, CA, NAG, FUC, MAN
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3-Quinoline Carboxamides Inhibitors Of Pi3K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2016-08-03 Classification: TRANSFERASE Ligands: 3QH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: 3QH, SO4
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Tankyrase In Complex With Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-05-13 Classification: TRANSFERASE/INHIBITOR Ligands: GOL, 3J1, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: GOL, 3J1, ZN
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Human Tankyrase 1 With Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-05-13 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, 3J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: ZN, 3J5
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Crystal Structure Of Tyrosine Kinase 2 Jh2 (Pseudo Kinase Domain) Complexed With Bms-066 Aka 2-Methoxy-N-({6-[3-Methyl-7-(Methylamino)-3,5,8,10-Tetraazatricyclo[7.3.0.0, 6]Dodeca-1(9),2(6),4,7,11-Pentaen-11-Yl]Pyridin-2-Yl}Methy L)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-03-18 Classification: TRANSFERASE/INHIBITOR Ligands: 3SM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3SM, SO4
