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Search Count: 12

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6C1S image
Phosphoinositide 3-Kinase Gamma Bound To An Pyrrolopyridinone Inhibitor

4YTC image
Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease

4YTF image
Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases

4YTH image
Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases

4YTI image
Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease

3JY9 image
Janus Kinase 2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2009-12-01
Classification: TRANSFERASE
Ligands: JZH, NA

3KCK image
A Novel Chemotype Of Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2009-11-24
Classification: TRANSFERASE
Ligands: 3KC

3IO7 image
2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2009-11-10
Classification: TRANSFERASE
Ligands: 1P5

3IOK image
2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2009-11-10
Classification: TRANSFERASE
Ligands: 1P6

3BGP image
Human Pim-1 Complexed With A Benzoisoxazole Inhibitor Vx1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2007-12-11
Classification: TRANSFERASE
Ligands: VX1

3BGQ image
Human Pim-1 Kinase In Complex With An Triazolo Pyridazine Inhibitor Vx2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2007-12-11
Classification: TRANSFERASE
Ligands: VX2

3BGZ image
Human Pim-1 Kinase In Complex With Diphenyl Indole Inhibitor Vx3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2007-12-11
Classification: TRANSFERASE
Ligands: VX3
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