Search Count: 12
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Phosphoinositide 3-Kinase Gamma Bound To An Pyrrolopyridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2018-06-27 Classification: Transferase/Transferase Inhibitor Ligands: EFV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: EFV, SO4
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 4HW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 4HW
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 4HZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 4HZ
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: 467 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 467
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Discovery Of Vx-509 (Decernotinib): A Potent And Selective Janus Kinase (Jak) 3 Inhibitor For The Treatment Of Autoimmune Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2015-08-12 Classification: Transferase/Transferase Inhibitor Ligands: VJK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: VJK
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Janus Kinase 2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-12-01 Classification: TRANSFERASE Ligands: JZH, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-01
Ligands: JZH, NA
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A Novel Chemotype Of Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-11-24 Classification: TRANSFERASE Ligands: 3KC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-24
Ligands: 3KC
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P5
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P6
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Human Pim-1 Complexed With A Benzoisoxazole Inhibitor Vx1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2007-12-11 Classification: TRANSFERASE Ligands: VX1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: VX1
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Human Pim-1 Kinase In Complex With An Triazolo Pyridazine Inhibitor Vx2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-12-11 Classification: TRANSFERASE Ligands: VX2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: VX2
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Human Pim-1 Kinase In Complex With Diphenyl Indole Inhibitor Vx3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-12-11 Classification: TRANSFERASE Ligands: VX3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: VX3
