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9Z1L image
Structure Of Kit V654A Mutant With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.54 Å Release Date: 2026-03-18
Classification: TRANSFERASE
Ligands: MRD, A1CZZ

9Z2S image
Structure Of Kit V654A Mutant With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2026-03-18
Classification: TRANSFERASE
Ligands: DMS, EDO, A1CZ3

8D73 image
Crystal Structure Of Egfr Lrtm With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.17 Å Release Date: 2022-07-27
Classification: SIGNALING PROTEIN
Ligands: GOL, QCR

8D76 image
Crystal Structure Of Egfr Lrtm With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2022-07-27
Classification: SIGNALING PROTEIN
Ligands: GOL, QFO

5JUN image
Pb2 Bound To An Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.69 Å Release Date: 2017-05-17
Classification: RNA BINDING PROTEIN
Ligands: 6NU

5JUR image
Pb2 Bound To An Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.93 Å Release Date: 2017-03-01
Classification: RNA BINDING PROTEIN
Ligands: 6NS

5F79 image
Influenza Pb2 Bound To An Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2016-12-07
Classification: Transcription/Inhibitor
Ligands: 4V7

5J40 image
The X-Ray Structure Of Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Resolution:2.17 Å Release Date: 2016-07-20
Classification: HYDROLASE/INHIBITOR
Ligands: ZN, MES, SO4

5J47 image
The X-Ray Structure Of Inhibitor Bound To Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Resolution:1.99 Å Release Date: 2016-07-20
Classification: HYDROLASE/INHIBITOR
Ligands: ZN, MES, 6JJ

5J4V image
The Crystal Structure Of Inhibitor Bound To Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Resolution:2.94 Å Release Date: 2016-07-20
Classification: HYDROLASE/INHIBITOR
Ligands: ZN, MES, SO4, 6JH

5J4Y image
The Crystal Structure Of N-(4-(2-(Thiazolo[5,4-C]Pyridin-2-Yl)Phenoxy)Phenyl)Acetamide Bound To Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Resolution:2.59 Å Release Date: 2016-07-20
Classification: HYDROLASE/INHIBITOR
Ligands: ZN, MES, SO4, 6JG

5BUH image
Influenza Pb2 Bound To A Hydroxymethyl Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2016-06-08
Classification: IMMUNE SYSTEM
Ligands: 4V7

4YD0 image
Influenza Polymerase Basic Protein 2 (Pb2) Bound To An Azaindole-Tetrazole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.62 Å Release Date: 2015-04-15
Classification: TRANSCRIPTION/INHIBITOR
Ligands: 4EW

4P8O image
S. Aureus Gyrase Bound To An Aminobenzimidazole Urea Inhibitor
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2014-10-29
Classification: ISOMERASE
Ligands: 883

4NCE image
Influenza Polymerase Basic Protein 2 (Pb2) Bound To 7-Methyl-Gtp
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2014-07-30
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: MGT, 11H

4NCM image
Influenza Polymerase Basic Protein 2 (Pb2) Bound To A Small-Molecule Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.82 Å Release Date: 2014-07-30
Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR
Ligands: 704

4P1U image
Influenza A (Flu) Virus Polymerase Basic Protein 2 (Pb2) Bound To Vx787, An Azaindole Inhibitor
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Resolution:2.52 Å Release Date: 2014-07-30
Classification: transferase/transferase inhibitor
Ligands: 21G

3B92 image
Novel Thio-Based Tace Inhibitors Part 2: Rational Design, Synthesis And Sar Of Thiol-Contaning Aryl Sufones
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2007-12-18
Classification: HYDROLASE
Ligands: ZN, 440

2OI0 image
Crystal Structure Analysis 0F The Tnf-A Coverting Enzyme (Tace) In Complexed With Aryl-Sulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2007-11-27
Classification: HYDROLASE
Ligands: ZN, 283

1QTI image
Acetylcholinesterase (E.C.3.1.1.7)
Organism: Torpedo californica
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 1999-12-29
Classification: HYDROLASE
Ligands: GNT
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