Search Count: 28
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Crystal Structure Of Egfr Exon20 Insertion Mutant In Complex With Enozertinib (Oric-114)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2025-11-12 Classification: SIGNALING PROTEIN Ligands: A1L8T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1L8T
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Discovery Of M5049: A Novel Selective Tlr7/8 Inhibitor For Treatment Of Autoimmunity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2020-12-30 Classification: IMMUNE SYSTEM Ligands: NAG, QLH, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: NAG, QLH, FMT
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Btk In Complex With Gdc-0834
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 2VL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 2VL, EDO, GOL
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Structure Of Btk With Rn486
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 7G6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7G6
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Btk1 Cocrystallized With Rn983
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 7G7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7G7
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Btk1 Soaked With Ibrutinib-Rev
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 1E8, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 1E8, DMS
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Btk1 Cocrystallized With Ibrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.08 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8E8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8E8
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Crystal Structure Of Btk With Cnx 774
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 7G8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7G8
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Btk1 In Complex With Cc 292
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 7G9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7G9
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Btk1 Binds Covalently To Hy-15771 Ono-4059
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 7GB, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7GB, DMS
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Crystal Structure Of Fat Domain Of Focal Adhesion Kinase (Fak) Bound To The Transcription Factor Mef2C
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2016-07-13 Classification: Transcription, protein binding |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
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Crystal Structure Of Yeast 20S Proteasome In Complex With Enone Carmaphycin Analogue 6
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-07-02 Classification: Hydrolase/Hydrolase Inhibitor Ligands: EC6 |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-07-02
Ligands: EC6
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Crystal Structure Of Yeast 20S Proteasome In Complex With Vinylketone Carmaphycin Analogue Vnk1
Organism: Saccharomyces cerevisiae s288c, Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-01-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ONK, VNK |
Organism: Saccharomyces cerevisiae s288c, Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
Ligands: ONK, VNK
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Crystal Structure Of Yeast 20S Proteasome In Complex With Epoxyketone Carmaphycin Analogue 3
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-01-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: OV2 |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
Ligands: OV2
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Crystal Structure Of Yeast 20S Proteasome In Complex With The Natural Product Carmaphycin A
Organism: Saccharomyces cerevisiae, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-01-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: OV1 |
Organism: Saccharomyces cerevisiae, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
Ligands: OV1
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Structure Of Porcine Pancreatic Elastase In 95% Acetone
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-04-18 Classification: HYDROLASE Ligands: CA, SO4, ACN |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2006-04-18
Ligands: CA, SO4, ACN
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Structure Of Porcine Pancreatic Elastase In 40/50/10 % Benzene
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-04-18 Classification: HYDROLASE Ligands: CA, SO4, IPA |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2006-04-18
Ligands: CA, SO4, IPA
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Structure Of Porcine Pancreatic Elastase In 40/50/10 Cyclohexane
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-04-18 Classification: HYDROLASE Ligands: CA, SO4, IPA |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2006-04-18
Ligands: CA, SO4, IPA
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Structure Of Porcine Pancreatic Elastase In 55% Dimethylformamide
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-04-18 Classification: HYDROLASE Ligands: CA, SO4, DMF |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2006-04-18
Ligands: CA, SO4, DMF
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Structure Of Porcine Pancreatic Elastase In 80% Ethanol
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-04-18 Classification: HYDROLASE Ligands: CA, SO4, EOH |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2006-04-18
Ligands: CA, SO4, EOH
