Search Count: 14
 |
C-Terminal Bromodomain Of Human Brd2 With 5-(1-Benzyl-4-Chloro-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, PE4, A1IBV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, PE4, A1IBV
 |
N-Terminal Bromodomain Of Human Brd4 With (5-(4-Chloro-1-((Tetrahydro-2H-Pyran-4-Yl)Methyl)-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, A1IB5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, A1IB5
 |
N-Terminal Bromodomain Of Human Brd4 With I-Bet567
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2022-12-14 Classification: TRANSCRIPTION Ligands: AKQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: AKQ, EDO
 |
C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-3-Methyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, P4M, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, P4M, MES
 |
C-Terminal Bromodomain Of Human Brd2 With (R)-7-((R)-1,2-Dihydroxyethyl)-1,3-Dimethyl-5-(1-Methyl-1H-Pyrazol-4-Yl)-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, 7PE, P4X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, 7PE, P4X
 |
C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, PE4, P0U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, PE4, P0U
 |
C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, PE4, P3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, PE4, P3R
 |
N-Terminal Bromodomain Of Human Brd2 With 5-(4-(4-Fluorophenyl)-1H-Imidazol-5-Yl)-1-Methylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-02-19 Classification: TRANSCRIPTION Ligands: SO4, NUQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-19
Ligands: SO4, NUQ, EDO
 |
N-Terminal Bromodomain Of Human Brd4 With 1-((1-Acetylpiperidin-4-Yl)Methyl)-2-(4-Hydroxy-3,5-Dimethylphenyl)-N-Methyl-1H-Benzo[D]Imidazole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: NUW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: NUW, EDO
 |
N-Terminal Bromodomain Of Human Brd4 With 1,3-Dimethyl-5-(1-((Tetrahydro-2H-Pyran-4-Yl)Methyl)-1H-Benzo[D]Imidazol-2-Yl)Pyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: EDO, NUB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: EDO, NUB
 |
N-Terminal Bromodomain Of Human Brd4 With 5-(1-(1,3-Dimethoxypropan-2-Yl)-5-Morpholino-1H-Benzo[D]Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: EDO, NV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: EDO, NV2
 |
N-Terminal Bromodomain Of Human Brd4 With 5-(1-(1,3-Dimethoxypropan-2-Yl)-5-Morpholino-1H-Benzo[D]Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: SO4, NUH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: SO4, NUH, EDO
 |
Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk147
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3YZ
 |
Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk199
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.29 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3Z0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3Z0