Search Count: 14
![]() |
Pi3Kg In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2019-01-30 Classification: TRANSFERASE Ligands: DD8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-30
Ligands: DD8
![]() |
Igfr-1R Complex With A Pyrimidine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-10-19 Classification: TRANSFERASE Ligands: GD5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-19
Ligands: GD5
![]() |
Igfr-1R Complex With A Pyrimidine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-10-19 Classification: TRANSFERASE Ligands: 8LN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-19
Ligands: 8LN
![]() |
Igfr-1R Complex With A Pyrimidine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-10-19 Classification: TRANSFERASE Ligands: ACT, OZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-19
Ligands: ACT, OZN
![]() |
Pkb Alpha In Complex With Azd5363
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2013-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0XZ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 0XZ, GOL
![]() |
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, YDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, YDI
![]() |
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, GOL, YDK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, GOL, YDK
![]() |
Synthesis And Evaluation Of Triazolones As Checkpoint Kinase 1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2012-03-14 Classification: TRANSFERASE Ligands: TQ1, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: TQ1, SO4, EDO
![]() |
Synthesis And Evaluation Of Triazolones As Checkpoint Kinase 1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2012-03-14 Classification: TRANSFERASE Ligands: GOL, YEX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: GOL, YEX, SO4
![]() |
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2012-01-25 Classification: TRANSFERASE Ligands: YDJ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: YDJ, PO4
![]() |
Jnk1 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, CFK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: SO4, CFK
![]() |
Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-08-11 Classification: TRANSFERASE Ligands: X8D, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: X8D, SO4
![]() |
Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-08-11 Classification: TRANSFERASE Ligands: X8E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: X8E, SO4
![]() |
Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2010-08-11 Classification: TRANSFERASE Ligands: X8I, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: X8I, SO4, GOL
