Search Count: 32
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Crystal Structure Of Human Haspin (Gsg2) Kinase Bound To Mu1963
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2024-10-16 Classification: TRANSFERASE Ligands: NI, MPD, A1IDE, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: NI, MPD, A1IDE, NA
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Crystal Structure Of Haspin (Gsg2) In Complex With Mu1464
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2024-09-11 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
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Crystal Structure Of Haspin (Gsg2) In Complex With Mu1668
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2024-09-11 Classification: TRANSFERASE Ligands: A1IDA, MPD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
Ligands: A1IDA, MPD, GOL
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Crystal Structure Of Human Haspin (Gsg2) Kinase Bound To Mu2181
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2024-09-11 Classification: TRANSFERASE Ligands: NI, A1IDC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
Ligands: NI, A1IDC
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Crystal Structure Of Human Haspin (Gsg2) Kinase Bound To Mu1959
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-09-11 Classification: TRANSFERASE Ligands: EPE, MPD, NA, A1IDD, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
Ligands: EPE, MPD, NA, A1IDD, NI
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Crystal Structure Of Human Haspin (Gsg2) Kinase Bound To Chemical Probe Mu1920
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2024-09-11 Classification: TRANSFERASE Ligands: A1IDF, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
Ligands: A1IDF, NI
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Crystal Structure Of Ck1 Delta In Complex With Pk-09-82
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-01-18 Classification: TRANSFERASE Ligands: SO4, EDO, EZQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, EDO, EZQ
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Crystal Structure Of Ck1 Delta In Complex With Vn725
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-01-18 Classification: TRANSFERASE Ligands: SO4, EDO, EYI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, EDO, EYI
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Crystal Structure Of Ck1 Delta In Complex With Pk-09-129
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2023-01-18 Classification: TRANSFERASE Ligands: SO4, EX9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, EX9
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Crystal Structure Of Hipk2 In Complex With Mu135 (Compound 21E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2021-03-03 Classification: TRANSFERASE Ligands: U82 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: U82
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Crystal Structure Of Clk1 In Complex With Furanopyrimidin Vn412
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: EDO, GOL, H3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: EDO, GOL, H3N
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Crystal Structure Of Clk1 In Complexed With Furo[3,2-B]Pyridine Compound 12H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-01-09 Classification: TRANSFERASE Ligands: H3E, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-09
Ligands: H3E, EDO
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Crystal Structure Of Clk1 In Complexed With Furo[3,2-B]Pyridine Compound Vn345 (Derivative Of Compound 12H)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-01-09 Classification: TRANSFERASE Ligands: GOL, H3H, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-09
Ligands: GOL, H3H, PO4
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Crystal Structure Of Clk1 In Complexed With Furo[3,2-B]Pyridine Compound Vn316 (Derivative Of Compound 12H)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2019-01-09 Classification: TRANSFERASE Ligands: PO4, H3Q, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-09
Ligands: PO4, H3Q, GOL
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Structure Of Phopsho-Cdk2-Cyclin A In Complex With An Atp-Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-01-25 Classification: TRANSFERASE Ligands: 6ZK, SGM, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 6ZK, SGM, MG
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Discovery Of Pyrazolo[1,5A]Pyrimidine-Based Pim1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-09-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 26K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 26K
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Discovery Of Pyrazolo[1,5A]Pyrimidine-Based Pim1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-09-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 26L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: 26L
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X-Ray Crystal Structure Of Compound 22K Bound To Human Chk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: 22K
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X-Ray Crystal Structure Of Compound 17R Bound To Human Chk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MI5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: MI5, GOL
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Crystal Structure Of Cyclin-Dependent Kinase 2 With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-01-22 Classification: TRANSFERASE Ligands: SC8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-22
Ligands: SC8
