Search Count: 14
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Crystal Structure Of The Catalytic Domain Of Human Pkc Alpha (D463N, V568I, S657E) In Complex With Nvp-Cjl037 At 2.48-A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2024-01-24 Classification: TRANSFERASE/INHIBITOR Ligands: V5U, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: V5U, MG
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Crystal Structure Of The Catalytic Domain Of Human Pkc Alpha (D463N, V568I, S657E) In Complex With Darovasertib (Nvp-Lxs196) At 2.82-A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2024-01-24 Classification: TRANSFERASE/INHIBITOR Ligands: W39 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: W39
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Tno155
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: VKS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: VKS, PO4
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: VKP, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: VKP, PO4
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Crystal Structure Of Human Nampt In Complex With Nvp-Ltm976
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2019-12-04 Classification: TRANSFERASE Ligands: OE4, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: OE4, PO4
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Crystal Structure Of Human Nampt In Complex With Nvp-Loq594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-10-03 Classification: TRANSFERASE Ligands: CVP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-03
Ligands: CVP
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Crystal Structure Of Human Nampt In Complex With Nvp-Lvr596
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2018-10-03 Classification: TRANSFERASE Ligands: CVJ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-03
Ligands: CVJ, PO4
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Crystal Structure Of Human Nampt In Complex With Nvp-Lod812
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-09-12 Classification: TRANSFERASE Ligands: BWA, GOL, PO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: BWA, GOL, PO4, DMS
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Crystal Structure Of Human Nampt In Complex With Nvp-Lqn520
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-09-12 Classification: TRANSFERASE Ligands: C5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: C5V
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-07-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 5OA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 5OA, PO4
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp099
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-06-29 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 5OD, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 5OD, PO4
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Tankyrase-1 Complexed With Small Molecule Inhibitor N-[(4-Oxo-3,4-Dihydroquinazolin-2-Yl)Methyl]-3-Phenyl-N-(Thiophen-2-Ylmethyl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-08-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SO4, 1XO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: ZN, SO4, 1XO
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Tankyrase-1 Complexed With Small Molecule Inhibitor 4-Chloro-5-Cyano-N-{2-[4-(4-Fluorobenzoyl)Piperidin-1-Yl]Ethyl}-2-Methoxybenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-08-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, NA, 1XP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: SO4, NA, 1XP
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Tankyrase-1 Complexed With Small Molecule Inhibitor 2-[4-(4-Fluorobenzoyl)Piperidin-1-Yl]-N-[(4-Oxo-3,5,7,8-Tetrahydro-4H-Pyrano[4,3-D]Pyrimidin-2-Yl)Methyl]-N-(Thiophen-2-Ylmethyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2013-08-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 1XQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: ZN, 1XQ, SO4