Search Count: 19
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Egfr Exon20 Insertion Mutant Asv Bound With (S)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN,TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1IMS, CL, EDO, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1IMS, CL, EDO, GOL, PEG
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Egfr Exon20 Insertion Mutant Svd Bound With (S)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN,TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1IMS, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1IMS, EDO, GOL
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Egfr Exon20 Insertion Mutant Svd Bound With Stx-721
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN,TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1A4E, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1A4E, CL, EDO, GOL
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Wildtype Egfr Bound With (R)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.12 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN Ligands: A1ILZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1ILZ
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Egfr Exon20 Insertion Mutant Npg Bound With (S)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2025-05-14 Classification: TRANSFERASE Ligands: A1IMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1IMS
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Egfr Exon20 Insertion Mutant Npg Bound With Stx-721
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2025-05-14 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
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Wild-Type Egfr Bound With Stx-721
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2025-05-14 Classification: TRANSFERASE Ligands: CL, A1IMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: CL, A1IMT
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Egfr Exon20 Insertion Mutant Npg Bound With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2025-01-29 Classification: TRANSFERASE Ligands: A1IEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: A1IEZ
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Egfr Exon20 Insertion Mutant Npg Bound With Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2025-01-29 Classification: TRANSFERASE Ligands: EDO, A1IE0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: EDO, A1IE0
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Wildtype Egfr Bound With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2025-01-29 Classification: ONCOPROTEIN Ligands: DTT, A1IEZ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: DTT, A1IEZ, CL
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Idh1 R132H Mutant In Complex With Idh305
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2017-11-08 Classification: OXIDOREDUCTASE Ligands: NDP, C81, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-08
Ligands: NDP, C81, FLC
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Idh1 R132H In Complex With Idh146
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-02-08 Classification: OXIDOREDUCTASE Ligands: NDP, 70Q, SO4, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: NDP, 70Q, SO4, EDO, DMS
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Idh1 R132H In Complex With Idh125
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2017-02-08 Classification: OXIDOREDUCTASE Ligands: NDP, 70P, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: NDP, 70P, FLC
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Structure Of Idh2 Mutant R172K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-02-08 Classification: OXIDOREDUCTASE Ligands: NDP, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: NDP, PEG
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Structure Of Idh2 Mutant R140Q
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2017-02-08 Classification: OXIDOREDUCTASE Ligands: NAP, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: NAP, EPE
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Idh1 R132H Mutant In Complex With Idh889
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-01-25 Classification: OXIDOREDUCTASE Ligands: FLC, 7J2, NDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: FLC, 7J2, NDP
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Crystal Structure Of Prmt5:Mep50 In Complex With Mta And H4 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2016-02-24 Classification: TRANSFERASE/PROTEIN BINDING Ligands: MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: MTA
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Heat Shock Protein 70 Substrate Binding Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2015-01-14 Classification: CHAPERONE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-14
Ligands: GOL
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Heat Shock Protein 70 Substrate Binding Domain With Covalently Linked Novolactone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2015-01-14 Classification: chaperone/chaperone inhibitor Ligands: 3UM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-14
Ligands: 3UM
