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Search Count: 6

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9GJQ image
Crystal Structure Of Humanised Cereblon From Magnetospirillum Gryphiswaldense Bound By Dihydrouracil-Indole Compound [1-(1H-Indol-6-Yl)Dihydro-2,4(1H,3H)-Pyrimidinedione].
Organism: Magnetospirillum gryphiswaldense
Method: X-RAY DIFFRACTION
Resolution:1.39 Å Release Date: 2025-09-03
Classification: LIGASE
Ligands: A1IMN, ZN

9ETQ image
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.59 Å Release Date: 2024-12-04
Classification: TRANSFERASE
Ligands: A1H63, SO4

9ETR image
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.82 Å Release Date: 2024-12-04
Classification: TRANSFERASE
Ligands: A1H64, SO4

7ONR image
Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKW, SO4

7ONS image
Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKT, SO4

7ONT image
Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKQ, SO4
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