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4DCB image
Y. Pestis Plasminogen Activator Pla In Complex With Human Plasminogen Activation Loop Peptide Alp11

3U73 image
Crystal Structure Of Stabilized Human Upar Mutant In Complex With Atf

4K24 image
Structure Of Anti-Upar Fab Atn-658 In Complex With Upar

3LAQ image
Structure-Based Engineering Of Species Selectivity In The Upa-Upar Interaction

4GLY image
Human Urokinase-Type Plasminogen Activator Upa In Complex With The Two-Disulfide Bridge Peptide Uk504

4JK5 image
Human Urokinase-Type Plasminogen Activator (Upa) In Complex With A Bicyclic Peptide Inhibitor (Uk18-D-Ser)

4JK6 image
Human Urokinase-Type Plasminogen Activator (Upa) In Complex With A Bicyclic Peptide Inhibitor (Uk18-D-Aba)

3IG6 image
Low Molecular Weigth Human Urokinase Type Plasminogen Activator 2-[6-(3'-Aminomethyl-Biphenyl-3-Yloxy)-4-(3-Dimethylamino-Pyrrolidin-1-Yl)-3,5-Difluoro-Pyridin-2-Yloxy]-4-Dimethylamino-Benzoic Acid Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2009-10-13
Classification: HYDROLASE
Ligands: 438, PO4

2VIW image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, D56

2VIP image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, SO4, L1R

2VIV image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, VG2

2VIQ image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, D55

2VIO image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, L1O

2VIN image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, SO4, 505

1URK image
Solution Structure Of The Amino Terminal Fragment Of Urokinase-Type Plasminogen Activator

3BT2 image
Structure Of Urokinase Receptor, Urokinase And Vitronectin Complex

3BT1 image
Structure Of Urokinase Receptor, Urokinase And Vitronectin Complex

3KID image
The Crystal Structures Of 2-Aminobenzothiazole-Based Inhibitors In Complexes With Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.71 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 2BS

3KGP image
Crystal Structures Of Urokinase-Type Plasminogen Activator In Complex With 4-(Aminomethyl) Benzoic Acid And 4-(Aminomethyl-Phenyl)-Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 4AZ, SO4

3KHV image
Crystal Structures Of Urokinase-Type Plasminogen Activator In Complex With 4-(Aminomethyl) Benzoic Acid And 4-(Aminomethyl-Phenyl)-Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 4AL, SO4, PGE
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