Structural Entry Filters:

Search Count: 42

4DCB image
Y. Pestis Plasminogen Activator Pla In Complex With Human Plasminogen Activation Loop Peptide Alp11
Organism: Yersinia pestis, Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2012-06-06
Classification: HYDROLASE
Ligands: MRD, MPD, C8E, PO4

3LAQ image
Structure-Based Engineering Of Species Selectivity In The Upa-Upar Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:3.20 Å Release Date: 2010-02-02
Classification: Hydrolase/Hydrolase Receptor
Ligands: NAG

3IG6 image
Low Molecular Weigth Human Urokinase Type Plasminogen Activator 2-[6-(3'-Aminomethyl-Biphenyl-3-Yloxy)-4-(3-Dimethylamino-Pyrrolidin-1-Yl)-3,5-Difluoro-Pyridin-2-Yloxy]-4-Dimethylamino-Benzoic Acid Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2009-10-13
Classification: HYDROLASE
Ligands: 438, PO4

2VIW image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, D56

2VIQ image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, D55

2VIN image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, SO4, 505

2VIO image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, L1O

2VIP image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, SO4, L1R

2VIV image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, VG2

1URK image
Solution Structure Of The Amino Terminal Fragment Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 1995-05-08
Classification: PLASMINOGEN ACTIVATION
Ligands: FUC

3BT1 image
Structure Of Urokinase Receptor, Urokinase And Vitronectin Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2008-03-25
Classification: IMMUNE SYSTEM
Ligands: NAG

3BT2 image
Structure Of Urokinase Receptor, Urokinase And Vitronectin Complex
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2008-03-25
Classification: IMMUNE SYSTEM
Ligands: NAG

3KID image
The Crystal Structures Of 2-Aminobenzothiazole-Based Inhibitors In Complexes With Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.71 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 2BS

3KGP image
Crystal Structures Of Urokinase-Type Plasminogen Activator In Complex With 4-(Aminomethyl) Benzoic Acid And 4-(Aminomethyl-Phenyl)-Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 4AZ, SO4

3KHV image
Crystal Structures Of Urokinase-Type Plasminogen Activator In Complex With 4-(Aminomethyl) Benzoic Acid And 4-(Aminomethyl-Phenyl)-Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 4AL, SO4, PGE

4H42 image
Synthesis Of A Weak Basic Upa Inhibitor And Crystal Structure Of Complex With Upa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.01 Å Release Date: 2013-10-30
Classification: HYDROLASE/INHIBITOR
Ligands: 11E, PG6

1TPG image
F1-G Module Pair Residues 1-91 (C83S) Of Tissue-Type Plasminogen Activator (T-Pa) (Nmr, 298K, Ph2.95, Representative Structure)
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 1995-09-15
Classification: PLASMINOGEN ACTIVATION

3LW2 image
Mouse Plasminogen Activator Inhibitor-1 (Pai-1)
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:1.93 Å Release Date: 2010-04-07
Classification: HYDROLASE INHIBITOR

3CVM image
High Resolution Structure Of A Stable Plasminogen Activator Inhibitor Type-1 In Its Protease Cleaved Form
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.02 Å Release Date: 2008-08-19
Classification: BLOOD CLOTTING

4DVA image
The Crystal Structure Of Human Urokinase-Type Plasminogen Activator Catalytic Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2013-01-16
Classification: HYDROLASE
Ligands: SO4, P6G
Protein Functional Filters:
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