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1PKR image
The Structure Of Recombinant Plasminogen Kringle 1 And The Fibrin Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.48 Å Release Date: 1994-01-31
Classification: PLASMINOGEN
Ligands: CL

4DCB image
Y. Pestis Plasminogen Activator Pla In Complex With Human Plasminogen Activation Loop Peptide Alp11
Organism: Yersinia pestis, Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2012-06-06
Classification: HYDROLASE
Ligands: MRD, MPD, C8E, PO4

3LAQ image
Structure-Based Engineering Of Species Selectivity In The Upa-Upar Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:3.20 Å Release Date: 2010-02-02
Classification: Hydrolase/Hydrolase Receptor
Ligands: NAG

6OG4 image
Plasminogen Binding Group A Streptococcal M Protein
Organism: Homo sapiens, Streptococcus pyogenes
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2019-07-24
Classification: HYDROLASE/PROTEIN BINDING
Ligands: SO4

4GLY image
Human Urokinase-Type Plasminogen Activator Upa In Complex With The Two-Disulfide Bridge Peptide Uk504
Organism: Homo sapiens, Synthetic
Method: X-RAY DIFFRACTION
Resolution:1.52 Å Release Date: 2013-05-15
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: SO4, NA, CL, P6G, GOL

4JK5 image
Human Urokinase-Type Plasminogen Activator (Upa) In Complex With A Bicyclic Peptide Inhibitor (Uk18-D-Ser)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2013-07-17
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: SO4, CL, P6G, ZBR

4JK6 image
Human Urokinase-Type Plasminogen Activator (Upa) In Complex With A Bicyclic Peptide Inhibitor (Uk18-D-Aba)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2013-07-17
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: SO4, CL, P6G, ZBR

3IG6 image
Low Molecular Weigth Human Urokinase Type Plasminogen Activator 2-[6-(3'-Aminomethyl-Biphenyl-3-Yloxy)-4-(3-Dimethylamino-Pyrrolidin-1-Yl)-3,5-Difluoro-Pyridin-2-Yloxy]-4-Dimethylamino-Benzoic Acid Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2009-10-13
Classification: HYDROLASE
Ligands: 438, PO4

2VIQ image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, D55

2VIO image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, L1O

2VIP image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, SO4, L1R

2VIW image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, D56

2VIN image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, SO4, 505

2VIV image
Fragment-Based Discovery Of Mexiletine Derivatives As Orally Bioavailable Inhibitors Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2008-01-22
Classification: HYDROLASE
Ligands: ACT, VG2

1URK image
Solution Structure Of The Amino Terminal Fragment Of Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 1995-05-08
Classification: PLASMINOGEN ACTIVATION
Ligands: FUC

3KID image
The Crystal Structures Of 2-Aminobenzothiazole-Based Inhibitors In Complexes With Urokinase-Type Plasminogen Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.71 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 2BS

3KHV image
Crystal Structures Of Urokinase-Type Plasminogen Activator In Complex With 4-(Aminomethyl) Benzoic Acid And 4-(Aminomethyl-Phenyl)-Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 4AL, SO4, PGE

3KGP image
Crystal Structures Of Urokinase-Type Plasminogen Activator In Complex With 4-(Aminomethyl) Benzoic Acid And 4-(Aminomethyl-Phenyl)-Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2009-12-01
Classification: HYDROLASE
Ligands: 4AZ, SO4

1TPK image
Crystal Structure Of The Kringle-2 Domain Of Tissue Plasminogen Activator At 2.4-Angstroms Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 1992-07-15
Classification: PLASMINOGEN ACTIVATOR
Ligands: CL

3U73 image
Crystal Structure Of Stabilized Human Upar Mutant In Complex With Atf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.19 Å Release Date: 2012-04-18
Classification: HYDROLASE/HYDROLASE RECEPTOR
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