Search Count: 14
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Crystal Structure Of Jak3 With Gcl258
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-08-20 Classification: TRANSFERASE Ligands: A1JJU, PHU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-20
Ligands: A1JJU, PHU
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Human Jak3 Kinase Domain With 1-(4-((2-((1-Methyl-1H-Pyrazol-4-Yl)Amino)Quinazolin-8-Yl)Amino)Piperidin-1-Yl)Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2022-02-02 Classification: SIGNALING PROTEIN Ligands: 934, SO4, PHU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-02
Ligands: 934, SO4, PHU
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Crystal Structure Of Jak3 In Complex With Fm601 (Compound 10A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-12-02 Classification: TRANSFERASE Ligands: RQZ, PHU, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: RQZ, PHU, EDO
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Crystal Structure Of Jak3 In Complex With Fm587 (Compound 9A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-12-02 Classification: TRANSFERASE Ligands: RQT, PHU, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: RQT, PHU, EDO
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Crystal Structure Of Jak3 In Complex With Compound 10 (Fm475)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-06-27 Classification: TRANSFERASE Ligands: F3W, PHU, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: F3W, PHU, GOL, EDO
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Crystal Structure Of Jak3 In Complex With Compound 11 (Fm481)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-06-27 Classification: TRANSFERASE Ligands: F4B, PHU, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: F4B, PHU, EDO
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Crystal Structure Of Jak3 In Complex With Compound 20 (Fm484)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-06-27 Classification: TRANSFERASE Ligands: F48, PHU, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: F48, PHU, EDO
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Crystal Structure Of Jak3 In Complex With Compound 4 (Fm381)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2016-10-26 Classification: TRANSFERASE Ligands: 79T, PHU, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-26
Ligands: 79T, PHU, EDO
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Crystal Structure Of Jak3 In Complex With Compound 5 (Fm409)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-10-26 Classification: TRANSFERASE Ligands: PHU, EDO, 79R, 79S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-26
Ligands: PHU, EDO, 79R, 79S
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Jak3 Kinase Domain In Complex With 2-Phenoxy-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-1-Cyclopropyl-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-10-16 Classification: Transferase/Transferase Inhibitor Ligands: PHU, 1DT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-16
Ligands: PHU, 1DT
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-1,2,2-Trimethyl-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: PHU, 933 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: PHU, 933
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Calcium-Calmodulin Complexed With The Calmodulin Binding Domain From A Small Conductance Potassium Channel Splice Variant And Phenylurea
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2012-09-12 Classification: METAL TRANSPORT/CALCIUM BINDING PROTEIN Ligands: SO4, CA, GOL, PHU |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2012-09-12
Ligands: SO4, CA, GOL, PHU
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Crystal Structure Of A Small Conductance Potassium Channel Splice Variant Complexed With Calcium-Calmodulin
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-05-30 Classification: METAL BINDING PROTEIN Ligands: CA, PHU, GOL, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: CA, PHU, GOL, SO4
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Crystal Structure Of Neutrophil Gelatinase-Associated Lipocalin Ngal (C87S Mutant) In Complex With Fragment 1026, Phenylurea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2011-10-12 Classification: APOPTOSIS Ligands: PHU, SO4, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: PHU, SO4, CL, EDO
