Search Count: 58
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Gcn2 (Eif2Alpha Kinase 4, E2Ak4) In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-05-04 Classification: TRANSFERASE Ligands: G41, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: G41, DMS
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Gcn2 (Eif2Alpha Kinase 4, E2Ak4) In Complex With Compound 1 (Dovitinib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-03-02 Classification: TRANSFERASE Ligands: 38O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-02
Ligands: 38O
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Mertk Kinase Domain In Complex With Nps-1034
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4K
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Mertk Kinase Domain In Complex With Quinazoline-Based Inhbitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4E, SO4
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Mertk Kinase Domain In Complex With A Bisaminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4N
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Mertk Kinase Domain In Complex With Purine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Q
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Mertk Kinase Domain In Complex With A Type 2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4T
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Mertk Kinase Domain With Type 1.5 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4W
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Mertk Kinase Domain With Type 1 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Z
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Mertk Kinase Domain With Type 3 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S5E, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S5E, CL, EDO
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Crystal Structure Of Mertk In Complex With A Type 1.5 Aminopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2020-11-04 Classification: TRANSFERASE Ligands: R6K, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-04
Ligands: R6K, CL, EDO
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Crystal Structure Of Mertk Kinase Domain In Complex With Ldc1267
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2020-10-28 Classification: TRANSFERASE Ligands: R6H, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: R6H, CL
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Crystal Structure Of Mertk Kinase Domain In Complex With Merestinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2020-10-28 Classification: TRANSFERASE Ligands: L1X, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: L1X, CL
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Apo Crystal Structure Of The Mertk Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2020-10-28 Classification: TRANSFERASE Ligands: CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: CL
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Crystal Structure Of Mertk Kinase Domain In Complex With Gilteritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2020-10-28 Classification: TRANSFERASE Ligands: C6F, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: C6F, CL, DMS
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Crystal Structure Of Mertk Kinase Domain In Complex With Unc2025
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2020-10-28 Classification: TRANSFERASE Ligands: R6N, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: R6N, CL, DMS
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Crystal Structure Of Helicobacter Pylori Adhesin Laba
Organism: Helicobacter pylori
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2019-12-18 Classification: SUGAR BINDING PROTEIN |
Organism: Helicobacter pylori
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
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Human Kras In Complex With Darpin K13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2019-04-24 Classification: SIGNALING PROTEIN Ligands: GDP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: GDP, SO4
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Human Kras In Complex With Darpin K19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-04-24 Classification: SIGNALING PROTEIN Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: SO4
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Crystal Structure Of Human C-Kit Kinase Domain In Complex With Azd3229-Analogue (Compound 18)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2018-09-19 Classification: SIGNALING PROTEIN Ligands: F82 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: F82
