Search Count: 39
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Crystal Structure Of The Hect Domain Of Smurf 2 In Complex With Inhibitor 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-04-16 Classification: LIGASE Ligands: TJQ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-16
Ligands: TJQ, PO4
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Crystal Structure Of The Hect Domain Of Smurf 1 In Complex With Inhibitor 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2025-04-16 Classification: LIGASE Ligands: TJQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-16
Ligands: TJQ
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Crystal Structure Of The Hect Domain Of Smurf1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2025-04-16 Classification: LIGASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-16
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Crystal Structure Of Tead4 In Complex With Peptide 1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-03-15 Classification: TRANSCRIPTION Ligands: GOL, MYR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-03-15
Ligands: GOL, MYR
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Crystal Structure Of Human Wdr5 In Complex With Compound Wm662
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2023-01-11 Classification: ONCOPROTEIN Ligands: X8N, GOL, SO4, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-11
Ligands: X8N, GOL, SO4, PGE
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Kras G12C In Complex With Gdp And Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: MG, NZ6, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: MG, NZ6, GDP
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Kras G12C In Complex With Gdp And Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: MG, NZX, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: MG, NZX, GDP
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Krasg12C In Complex With Gdp And Jdq443
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2022-04-27 Classification: HYDROLASE Ligands: MG, H2T, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-27
Ligands: MG, H2T, GDP
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Krasg12C In Complex With Gdp And Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2022-04-27 Classification: HYDROLASE Ligands: MG, H40, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-27
Ligands: MG, H40, GDP
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Krasg12C In Complex With Gdp And Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-04-27 Classification: HYDROLASE Ligands: MG, H0O, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-27
Ligands: MG, H0O, GDP
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Pcsk9 In Complex With A Cyclic Peptide Ldlr Disruptor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-11-24 Classification: LIPID TRANSPORT, HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
Ligands: CA
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Pcsk9 In Complex With Pcsk9I A 13Mer Cyclic Peptide Ldlr Disruptor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-11-10 Classification: LIPID TRANSPORT, HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: CA
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X-Ray Structure Of Hdm2/Cmr19 At 1.45A: Discovery, X-Ray Structure And Cpp-Conjugation Enabled Uptake Of P53/Mdm2 Macrocyclic Peptide Inhibitors
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2021-09-22 Classification: LIGASE Ligands: SO4, CL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: SO4, CL
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 1: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HJW
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 2 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKE, CHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKE, CHD
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 4 At 2.2A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKZ
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 9 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HL8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HL8
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Apo Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Gnti-Deficient Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, MLI, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, MLI, CA
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Apo Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, EDO, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, EDO, CA
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Compound 2 Bound Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, M3D, EDO, CA, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, M3D, EDO, CA, TRS
