Search Count: 18
![]() |
Crystal Structure Of Human Syk In Complex With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-04-24 Classification: TRANSFERASE Ligands: A1H2W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-24
Ligands: A1H2W, GOL
![]() |
Crystal Structure Of Syk Kinase In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-04-24 Classification: TRANSFERASE Ligands: A1H2Y, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-24
Ligands: A1H2Y, GOL
![]() |
Crystal Structure Of The Legionella Pneumophila Chia C-Terminal Domain
Organism: Legionella pneumophila 130b
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2020-04-22 Classification: SUGAR BINDING PROTEIN Ligands: MPD, MRD |
Organism: Legionella pneumophila 130b
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: MPD, MRD
![]() |
The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7W |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: H7W
![]() |
The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With An Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7Z |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: H7Z
![]() |
Crystal Structure Of The Alk Kinase Domain In Complex With Entrectinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: YMX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: YMX
![]() |
Crystal Structure Of The Alk Kinase Domain In Complex With Cmpd 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: U4W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: U4W, GOL
![]() |
Structure Of Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: FSU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: FSU
![]() |
Structure Of Human Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: D7N
![]() |
Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: SO4, GOL, FSU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: SO4, GOL, FSU
![]() |
Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: D7N, SO4
![]() |
Structure Of Human Anaplastic Lymphoma Kinase In Complex With Nvp- Tae684
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-07-28 Classification: TRANSFERASE Ligands: GUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-28
Ligands: GUI
![]() |
Structure Of Human Anaplastic Lymphoma Kinase In Complex With Pha- E429
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-07-28 Classification: TRANSFERASE Ligands: 571 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-28
Ligands: 571
![]() |
Optimisation Of 6,6-Dimethyl Pyrrolo 3,4-C Pyrazoles: Identification Of Pha-793887, A Potent Cdk Inhibitor Suitable For Intravenous Dosing
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2010-02-23 Classification: CELL CYCLE Ligands: SO4, 889 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: SO4, 889
![]() |
Crystal Structure Of Gsk-3 Beta In Complex With Nms-869553A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-03-03 Classification: TRANSFERASE Ligands: 553 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-03
Ligands: 553
![]() |
Structure Of Cdk2-Cyclin A With Pha-630529
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2005-12-08 Classification: TRANSFERASE Ligands: 529, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-12-08
Ligands: 529, SO4
![]() |
Structure Of Cdk2 Complexed With Pnu-181227
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2004-06-17 Classification: TRANSFERASE Ligands: N5B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-06-17
Ligands: N5B
![]() |
Structure Of Cdk2/Cyclin A With Pnu-292137
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2004-06-10 Classification: TRANSFERASE Ligands: SO4, 292 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-06-10
Ligands: SO4, 292
