Search Count: 23
![]() |
Crystal Structure Of Cdk2/Cyclin E In Complex With Pf-06873600
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2021-06-23 Classification: CELL CYCLE Ligands: WG1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-23
Ligands: WG1
![]() |
Crystal Structure Of Pi3Kalpha Selective Inhibitor Pf-06843195
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VXY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VXY
![]() |
Crystal Structure Of Pi3Kalpha Selective Inhibitor 11-1575
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY4
![]() |
Crystal Structure Of Pi3Kalpha Inhibitor 10-5429
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY1
![]() |
Crystal Structure Of Pi3Kalpha Inhibitor 4-0686
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VYP
![]() |
Structure Of The Catalytic Domain Of Parp1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: SO4
![]() |
Structure Of The Catalytic Domain Of Parp1 In Complex With Talazoparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: 2YQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: 2YQ
![]() |
Structure Of The Catalytic Domain Of Parp1 In Complex With Olaparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: 09L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: 09L
![]() |
Structure Of The Catalytic Domain Of Parp1 In Complex With Niraparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: 3JD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: 3JD, SO4
![]() |
Structure Of The Catalytic Domain Of Parp1 In Complex With Veliparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: 78P, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: 78P, SO4
![]() |
Structure Of The Catalytic Domain Of Tankyrase 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: ZN
![]() |
Structure Of The Catalytic Domain Of Tankyrase 1 In Complex With Talazoparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: ZN, 2YQ, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: ZN, 2YQ, MES
![]() |
Structure Of The Catalytic Domain Of Tankyrase 1 In Complex With Olaparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: ZN, 09L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: ZN, 09L
![]() |
Structure Of The Catalytic Domain Of Tankyrase 1 In Complex With Niraparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: ZN, 3JD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: ZN, 3JD, SO4
![]() |
Structure Of The Catalytic Domain Of Tankyrase 1 In Complex With Veliparib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2021-01-06 Classification: TRANSFERASE Ligands: 78P, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: 78P, ZN
![]() |
Egfr (L858R, T790M, V948R) In Complex With N-{3-[(2-{[4-(4-Methylpiperazin-1-Yl)Phenyl]Amino}-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl)Oxy]Phenyl}Prop-2-Enamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 633, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 633, SO4, GOL
![]() |
Egfr (L858R, T790M, V948R) In Complex With N-[3-({2-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl}Oxy)Phenyl]Prop-2-Enamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 634, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 634, SO4, GOL
![]() |
Egfr (L858R, T790M, V948R) In Complex With 1-[(3R,4R)-3-[({2-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl}Oxy)Methyl]-4-(Trifluoromethyl)Pyrrolidin-1-Yl]Prop-2-En-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 63A, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 63A, SO4, GOL
![]() |
Egfr (L858R, T790M, V948R) In Complex With 1-{(3R,4R)-3-[5-Chloro-2-(1-Methyl-1H-Pyrazol-4-Ylamino)-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yloxymethyl]-4-Methoxy-Pyrrolidin-1-Yl}Propenone (Pf-06459988)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 630, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 630, SO4
![]() |
2-((1H-Benzo[D]Imidazol-1-Yl)Methyl)-4H-Pyrido[1,2-A]Pyrimidin-4-Ones As Novel Pkm2 Activators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: FBP, 1OX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: FBP, 1OX
