Structural Entry Filters:

Search Count: 12

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5DXH image
P110Alpha/P85Alpha With Compound 5

5DXT image
P110Alpha With Gdc-0326

5DXU image
P110Delta/P85Alpha With Gdc-0326

4J6I image
Discovery Of Thiazolobenzoxepin Pi3-Kinase Inhibitors That Spare The Pi3-Kinase Beta Isoform

4HLE image
Compound 21 (1-Alkyl-Substituted 1,2,4-Triazoles)

3T8M image
Rational Design Of Pi3K-Alpha Inhibitors That Exhibit Selectivity Over The Pi3K-Beta Isoform

3R7Q image
Structure-Based Design Of Thienobenzoxepin Inhibitors Of Pi3- Kinase

3R7R image
Structure-Based Design Of Thienobenzoxepin Inhibitors Of Pi3-Kinase

3NZS image
Structure-Based Optimization Of Pyrazolo -Pyrimidine And -Pyridine Inhibitors Of Pi3-Kinase

3NZU image
Structure-Based Optimization Of Pyrazolo -Pyrimidine And -Pyridine Inhibitors Of Pi3-Kinase

3DBS image
Structure Of Pi3K Gamma In Complex With Gdc0941
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2008-06-17
Classification: TRANSFERASE
Ligands: GD9

1YGC image
Short Factor Viia With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2005-01-18
Classification: HYDROLASE
Ligands: CA, SO4, 905
Protein Functional Filters:
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