Search Count: 18
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Crystal Structure Of Partially Phosphorylated Ret V804M Tyrosine Kinase Domain Complexed With Pdd00018412
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2020-03-11 Classification: ONCOPROTEIN Ligands: H6W, EDO, FMT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: H6W, EDO, FMT, CL
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Crystal Structure Of Phosphorylated Ret V804M Tyrosine Kinase Domain Complexed With Pdd00018366
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2020-03-11 Classification: ONCOPROTEIN Ligands: H72, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: H72, FMT
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Polyadpribosyl Glycohydrolase In Complex With Pdd00016690
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2018-11-14 Classification: HYDROLASE Ligands: DMS, GOL, SO4, 7JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: DMS, GOL, SO4, 7JC
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Polyadpribosyl Glycosidase In Complex With Pdd00017299
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-11-14 Classification: HYDROLASE Ligands: 73L, DMS, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: 73L, DMS, GOL, SO4
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Polyadpribosyl Glycohydrolase In Complex With Pdd00013907
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-11-14 Classification: HYDROLASE Ligands: DMS, GOL, 7JB, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: DMS, GOL, 7JB, SO4
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Polyadpribosyl Glycosidase In Complex With Pdd00014909
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2018-11-14 Classification: HYDROLASE Ligands: DMS, GOL, 70J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: DMS, GOL, 70J, SO4
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Crystal Structure Of Iso-Citrate Dehydrogenase R132H In Complex With A Novel Inhibitor (Compound 13A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-12-14 Classification: OXIDOREDUCTASE Ligands: NDP, 6N3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: NDP, 6N3
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Crystal Structure Of Iso-Citrate Dehydrogenase 1 [Idh1 (R132H)] In Complex With A Novel Inhibitor (Compound 2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2016-12-14 Classification: OXIDOREDUCTASE Ligands: NDP, 6MX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: NDP, 6MX
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Polyadpribosyl Glycosidase In Complex With Pdd00017262
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-10-12 Classification: HYDROLASE Ligands: 6WJ, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 6WJ, SO4, DMS
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Crystal Structure Of The Catalytic Domain Of Human Tyrosyl Dna Phosphodiesterase 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2016-05-04 Classification: HYDROLASE Ligands: MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: MG, GOL
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Crystal Structure Of The Catalytic Domain Of Human Tyrosyl Dna Phosphodiesterase 2 In Complex With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2016-05-04 Classification: HYDROLASE Ligands: 6FQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 6FQ
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Crystal Structure Of M2Htdp2-Cat In Complex With A Small Molecule Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-05-04 Classification: HYDROLASE Ligands: 6FQ, MG, GOL, EDO, ACT |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 6FQ, MG, GOL, EDO, ACT
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Crystal Structure Of M2Htdp2-Cat In Complex With A Small Molecule Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-05-04 Classification: HYDROLASE Ligands: 6FV, TLA, GOL, EDO, MN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 6FV, TLA, GOL, EDO, MN
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The Discovery Of 2-Substituted Phenol Quinazolines As Potent And Selective Ret Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2016-02-17 Classification: TRANSFERASE Ligands: DTQ, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-17
Ligands: DTQ, FMT
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Pkb Alpha In Complex With Azd5363
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2013-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0XZ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 0XZ, GOL
