Search Count: 20
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Co-Structure Of Human Glycogen Synthase Kinase Beta With 1-(6-((2-((6-Amino-5-Nitropyridin-2-Yl)Amino)Ethyl)Amino)-2-(2,4-Dichlorophenyl)Pyridin-3-Yl)-4-Methylpiperazin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2020-01-15 Classification: TRANSFERASE Ligands: QQA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: QQA, PO4
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Co-Structure Of Human Glycogen Synthase Kinase Beta With A Selective (5-Imidazol-2-Yl-4-Phenylpyrimidin-2-Yl)[2-(2-Pyridylamino)Ethyl]Amine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-11-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GOL, 65C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-08
Ligands: GOL, 65C
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Benzofuropyrimidinone Inhibitors Of Pim-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-01-16 Classification: TRANSFERASE Ligands: IMD, 79O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: IMD, 79O
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Benzofuropyrimidinone Inhibitors Of Pim-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2013-01-16 Classification: TRANSFERASE Ligands: IMD, R9P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: IMD, R9P
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Benzofuropyrimidinone Inhibitors Of Pim-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2013-01-16 Classification: TRANSFERASE Ligands: IMD, HY7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: IMD, HY7
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: EUI, ACP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: EUI, ACP, MG
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: MG, ATP, 5Y0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: MG, ATP, 5Y0
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: ACP, MG, 2P7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: ACP, MG, 2P7
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: YQY, ACP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: YQY, ACP, MG
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Aminoalkylpyrimidine Inhibitor Complexes With Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-11-21 Classification: TRANSFERASE Ligands: 3O4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-21
Ligands: 3O4
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Aminoalkylpyrimidine Inhibitor Complexes With Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-11-21 Classification: TRANSFERASE Ligands: O19 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-21
Ligands: O19
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Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-08-29 Classification: CHAPERONE Ligands: 99B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 99B
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Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2012-08-29 Classification: CHAPERONE Ligands: 99A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 99A
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Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-08-29 Classification: CHAPERONE Ligands: 592 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 592
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Complex Of The Ephb4 Kinase Domain With An Oxindole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2012-08-01 Classification: TRANSFERASE Ligands: 30K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-01
Ligands: 30K
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Complex Of Ck2 With A Cdc7 Inhibitor
Organism: Zea mays
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-05-23 Classification: TRANSFERASE Ligands: WUL |
Organism: Zea mays
Method: X-RAY DIFFRACTION
Release Date: 2012-05-23
Ligands: WUL
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Complexes Of Pi3Kgamma With Isoform Selective Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2012-05-09 Classification: TRANSFERASE Ligands: SO4, EM7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: SO4, EM7
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Complexes Of Pi3Kgamma With Isoform Selective Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2012-05-09 Classification: TRANSFERASE Ligands: SO4, 751 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: SO4, 751
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Complexes Of Pi3Kgamma With Isoform Selective Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2012-05-09 Classification: TRANSFERASE Ligands: SO4, O92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: SO4, O92
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Complexes Of Pi3Kgamma With Isoform Selective Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2012-05-09 Classification: TRANSFERASE Ligands: 534 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: 534
