Search Count: 11
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Prmt5 Bound To Compound 6 And Mta
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1CMW, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: A1CMW, MTA
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Prmt5 Bound To Compound 12 And Mta
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1CMZ, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: A1CMZ, MTA
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Prmt5 Bound To Compound 8 And Mta
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MTA, A1CM0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: MTA, A1CM0, SO4
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Mth1 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: S3O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: S3O
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Mth1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: 8JF
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Mth1 In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GN6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: GN6
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Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-09-19 Classification: TRANSFERASE/INHIBITOR Ligands: KK7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: KK7
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Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-09-19 Classification: TRANSFERASE/INHIBITOR Ligands: KK8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: KK8
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Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2018-09-19 Classification: TRANSFERASE/INHIBITOR Ligands: S0L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: S0L
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Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2017-11-29 Classification: Transferase/Transferase Inhibitor Ligands: YAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-29
Ligands: YAM
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Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-12-21 Classification: Transferase/Transferase Inhibitor Ligands: 7FM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: 7FM
