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Search Count: 11

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9PXZ image
Prmt5 Bound To Compound 6 And Mta
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.47 Å Release Date: 2026-01-07
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: A1CMW, MTA

9PY0 image
Prmt5 Bound To Compound 12 And Mta
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.36 Å Release Date: 2026-01-07
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: A1CMZ, MTA

9PY1 image
Prmt5 Bound To Compound 8 And Mta
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.04 Å Release Date: 2026-01-07
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: MTA, A1CM0, SO4

6US2 image
Mth1 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2020-04-01
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: S3O

6US3 image
Mth1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.47 Å Release Date: 2020-04-01
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: 8JF

6US4 image
Mth1 In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2020-04-01
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: GN6

6E2M image
Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.25 Å Release Date: 2018-09-19
Classification: TRANSFERASE/INHIBITOR
Ligands: KK7

6E2N image
Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2018-09-19
Classification: TRANSFERASE/INHIBITOR
Ligands: KK8

6E2O image
Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.39 Å Release Date: 2018-09-19
Classification: TRANSFERASE/INHIBITOR
Ligands: S0L

5TOB image
Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.12 Å Release Date: 2017-11-29
Classification: Transferase/Transferase Inhibitor
Ligands: YAM

5TO8 image
Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.98 Å Release Date: 2016-12-21
Classification: Transferase/Transferase Inhibitor
Ligands: 7FM
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