Search Count: 18
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7F9, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7F9, SO4
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-02-22 Classification: SIGNALING PROTEIN Ligands: 7FX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FX, SO4
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: TF3, 7F9, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: TF3, 7F9, MG
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FW, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FW, TF3, CL
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FV, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FV, TF3, CL
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Application Of Off-Rate Screening In The Identification Of Novel Pan-Isoform Inhibitors Of Pyruvate Dehydrogenase Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-02-22 Classification: TRANSFERASE Ligands: 7FE, TF3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7FE, TF3, CL
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, B21 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, B21
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, G14 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, G14
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, 4FF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, 4FF
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, 4G2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, 4G2
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 4F8, 12P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 4F8, 12P
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, 4FY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, 4FY
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, 4G8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, 4G8
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, 4G5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, 4G5
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-01-12 Classification: ISOMERASE Ligands: 12P, 4GE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 12P, 4GE
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Discovery Of Cell-Active Phenyl-Imidazole Pin1 Inhibitors By Structure-Guided Fragment Evolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-10-27 Classification: ISOMERASE Ligands: PE4, ODK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: PE4, ODK
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4,5 Diaryl Isoxazole Hsp90 Chaperone Inhibitors: Potential Therapeutic Agents For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-12-11 Classification: CHAPERONE Ligands: 2GJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: 2GJ
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4,5 Diaryl Isoxazole Hsp90 Chaperone Inhibitors: Potential Therapeutic Agents For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-12-11 Classification: CHAPERONE Ligands: 2EQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: 2EQ
