Search Count: 52
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Crystal Structure Of Flap Endonuclease Fen1 With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2025-09-24 Classification: HYDROLASE Ligands: MG, EDO, A1JD4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-24
Ligands: MG, EDO, A1JD4
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Crystal Structure Of Flap Endonuclease Fen1 With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2025-09-24 Classification: HYDROLASE Ligands: A1JED, TEW, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-24
Ligands: A1JED, TEW, MG
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ7
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ8, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ8, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ9
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: Q6K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: Q6K, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations. Compound 51 Bound To Egfrinsnpg [V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-02-05 Classification: SIGNALING PROTEIN Ligands: A1IUK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1IUK
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Estrogen Receptor Alpha In Complex With Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2023-02-01 Classification: TRANSCRIPTION Ligands: H09 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: H09
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-02-01 Classification: GENE REGULATION Ligands: GZI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: GZI
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Human Gls In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, 04A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, 04A
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Human Gls In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: R90 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: R90
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Human Gls In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, 5XX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, 5XX
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Human Gls In Complex With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2023-01-18 Classification: HYDROLASE Ligands: SO4, R0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: SO4, R0C
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Di-Methyl Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VJZ, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VJZ, CL, DMS
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Di-Methyl, Cyano Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VK2, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VK2, CL, DMS
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Tri-Methyl Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VK5, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VK5, CL
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Mertk Kinase Domain In Complex With Nps-1034
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4K
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Mertk Kinase Domain In Complex With Quinazoline-Based Inhbitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4E, SO4
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Mertk Kinase Domain In Complex With A Bisaminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4N
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Mertk Kinase Domain In Complex With Purine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Q
