Search Count: 17
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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B-Raf Wild-Type Kinase Domain In Complex With A Purinylpyridinylamino-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2016-05-04 Classification: Transferase/Transferase Inhibitor Ligands: 5XJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5XJ
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Human Gkrp Bound To Amg-2526 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-10-08 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TE, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 2TE, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0771 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TF, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TF, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-2668
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TG, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TG, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3227 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TJ, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TJ, S6P, IOD, GOL, SO4
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Gkrp Bound To Amg0556 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UW, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UW, S6P, IOD, GOL, SO4
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Gkrp Bound To Amg-0471 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UX, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UX, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-5112 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2UY, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2UY, S6P, IOD, GOL, SO4
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Human Gkrp Complexed To Amg-3969 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG9, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG9, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-5980 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG0, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG0, S6P, IOD, GOL, SO4
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Crystal Structure Of Human Pi3K-Gamma In Complex With Amg511
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-08-29 Classification: Transferase/Inhibitor Ligands: SO4, 14K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: SO4, 14K
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Crystal Structure Of Human Pi3K-Gamma In Complex With A Pyridyl-Triazine-Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2012-08-08 Classification: Transferase/Inhibitor Ligands: SO4, F1S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: SO4, F1S
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Crystal Structure Of Human Pi3K-Gamma In Complex With A Pyridyl-Triazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2012-05-16 Classification: Transferase/Inhibitor Ligands: SO4, 0KO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: SO4, 0KO
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Crystal Structure Of Pi3K-Gamma In Complex With A Quinoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2011-06-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 2NQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-08
Ligands: SO4, 2NQ
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Crystal Structure Of Dimeric Abscisic Acid (Aba) Receptor Pyrabactin Resistance 1 (Pyr1) With Aba-Bound Closed-Lid And Aba-Free Open-Lid Subunits
Organism: Arabidopsis thaliana
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2009-11-17 Classification: HORMONE RECEPTOR, SIGNALING PROTEIN Ligands: A8S |
Organism: Arabidopsis thaliana
Method: X-RAY DIFFRACTION
Release Date: 2009-11-17
Ligands: A8S
