Search Count: 17
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Blimp-1 With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2026-01-14 Classification: TRANSCRIPTION Ligands: A1CNQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-14
Ligands: A1CNQ
 |
Cereblon Ternary Complex With Blimp1 And Compound 5
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.20 Å Release Date: 2026-01-14 Classification: LIGASE Ligands: ZN, A1CN1 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-01-14
Ligands: ZN, A1CN1
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Cdk6 To Cdk4 Active Site Surrogate In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2025-12-17 Classification: TRANSFERASE/INHIBITOR Ligands: A1CIF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: A1CIF
 |
Cdk6 To Cdk4 Active Site Surrogate In Complex With Pf-07220060
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-12-17 Classification: TRANSFERASE/INHIBITOR Ligands: A1AZ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: A1AZ4
 |
Gsk3Beta In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2025-12-17 Classification: TRANSFERASE/INHIBITOR Ligands: A1CIF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: A1CIF
 |
Crystal Structure Of Cdk2/Cyclin E In Complex With Pf-06873600
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2021-06-23 Classification: CELL CYCLE Ligands: WG1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-23
Ligands: WG1
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 10B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: FKY
 |
Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 13B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GO7
 |
Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 19.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GOD
 |
Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GXA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: GXA
 |
Design And Synthesis Of A Novel Pyrrolidinyl Pyrido Pyrimidinone Derivative As A Potent Inhibitor Of Pi3Ka And Mtor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-04-03 Classification: Transferase/Transferase Inhibitor Ligands: 0TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-03
Ligands: 0TA
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Design And Synthesis Of A Novel Pyrrolidinyl Pyrido Pyrimidinone Derivative As A Potent Inhibitor Of Pi3Ka And Mtor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-04-03 Classification: Transferase/Transferase Inhibitor Ligands: 0TB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-03
Ligands: 0TB
 |
Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: WOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: WOE
 |
Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: FU5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: FU5
 |
Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: FU3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: FU3
 |
Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: FU7, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: FU7, PO4
 |
4-Methylpteridineones As Orally Active And Selective Pi3K/Mtor Dual Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2010-09-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OAW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-22
Ligands: OAW