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9VFO image
Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 2-Amino-N-(5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2026-04-22
Classification: TRANSFERASE
Ligands: A1ER0

9VGR image
Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 4-((5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Carbamoyl)-1-Methyl-3H-Pyrazol-1-Ium-3-Ide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2026-04-22
Classification: CYTOSOLIC PROTEIN
Ligands: A1ER9

9VIR image
Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor N-(5-((5-Chloro-4-(((3As,6R,6Ar)-6-Methoxy-3A,5,6,6A-Tetrahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-(((2R,7Ar)-2-Fluorotetrahydro-1H-Pyrrolizin-7A(5H)-Yl)Methoxy)Phenyl)-1-Methyl-1H-Pyrazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2026-04-22
Classification: CYTOSOLIC PROTEIN
Ligands: A1ESF

9UD7 image
Crystal Structure Of Human Glutaminyl Cyclase In Complex With Inhibitor Cl7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.49 Å Release Date: 2026-04-08
Classification: TRANSFERASE
Ligands: ZN, A1EOY, MG, GOL, TRS

22OZ image
Structural Insights Into Hpar-Mediated Recognition Of Hrpx And Hrpg In Xanthomonas Campestris Pv. Campestris

9V70 image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:2.82 Å Release Date: 2026-02-18
Classification: TRANSFERASE
Ligands: ADP, MG

9V71 image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:2.52 Å Release Date: 2026-02-18
Classification: TRANSFERASE
Ligands: ADP, MG

9V72 image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:2.76 Å Release Date: 2026-02-18
Classification: TRANSFERASE
Ligands: MG, ADP

9V7E image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2026-02-18
Classification: TRANSFERASE
Ligands: ADP, MG

9V73 image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:2.27 Å Release Date: 2026-01-28
Classification: TRANSFERASE
Ligands: ANP

9V79 image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:2.12 Å Release Date: 2026-01-28
Classification: TRANSFERASE
Ligands: MG, ANP

9WYQ image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2026-01-28
Classification: TRANSFERASE

9WYR image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2026-01-28
Classification: TRANSFERASE
Ligands: ATP, MG

9WYS image
Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION
Resolution:2.79 Å Release Date: 2026-01-28
Classification: TRANSFERASE
Ligands: ADP, MG

9KMB image
Crystal Structure Of Human Glutaminyl Cyclase In Complex With N-(2-(1H-Imidazol-5-Yl)Ethyl)-4-Methoxybenzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.28 Å Release Date: 2025-06-25
Classification: TRANSFERASE
Ligands: ZN, A1EFY

9ISD image
Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With The Inhibitor N-(1H-Benzo[D]Imidazol-5-Yl)-1-Phenylmethanesulfonamide (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.37 Å Release Date: 2025-03-12
Classification: TRANSFERASE
Ligands: ZN, A1D93, GOL, DMS, DMF, PEG

9IVV image
Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With The Inhibitor 3-((2-(1H-Imidazol-5-Yl)Ethyl)Carbamoyl)-4-Amino-1,2,5-Oxadiazole 2-Oxide (Compound 13)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.96 Å Release Date: 2025-03-12
Classification: TRANSFERASE
Ligands: ZN, A1D94, DMS, GOL, DMF

8XFV image
Crystal Structure Of Human Golgi Resident Glutaminyl Cyclase In Complex With (Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-(Piperidin-4-Yloxy)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.13 Å Release Date: 2024-06-12
Classification: TRANSFERASE
Ligands: ZN, A1D46

8XGA image
Crystal Structure Of Human Golgi Resident Glutaminyl Cyclase In Complex With (Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-((Tetrahydro-2H-Pyran-4-Yl)Oxy)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.54 Å Release Date: 2024-06-12
Classification: TRANSFERASE
Ligands: ZN, A1D47

8XGB image
Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With (S)-1-(1H-Benzo[D]Imidazol-5-Yl)-5-(4-Propoxyphenyl)Imidazolidin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.24 Å Release Date: 2024-06-12
Classification: TRANSFERASE
Ligands: ZN, A1D49
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