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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 2-Amino-N-(5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-04-22 Classification: TRANSFERASE Ligands: A1ER0 |
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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 4-((5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Carbamoyl)-1-Methyl-3H-Pyrazol-1-Ium-3-Ide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-22 Classification: CYTOSOLIC PROTEIN Ligands: A1ER9 |
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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor N-(5-((5-Chloro-4-(((3As,6R,6Ar)-6-Methoxy-3A,5,6,6A-Tetrahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-(((2R,7Ar)-2-Fluorotetrahydro-1H-Pyrrolizin-7A(5H)-Yl)Methoxy)Phenyl)-1-Methyl-1H-Pyrazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2026-04-22 Classification: CYTOSOLIC PROTEIN Ligands: A1ESF |
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Crystal Structure Of Human Glutaminyl Cyclase In Complex With Inhibitor Cl7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2026-04-08 Classification: TRANSFERASE Ligands: ZN, A1EOY, MG, GOL, TRS |
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Structural Insights Into Hpar-Mediated Recognition Of Hrpx And Hrpg In Xanthomonas Campestris Pv. Campestris
Organism: Xanthomonas campestris pv. campestris (strain atcc 33913 / dsm 3586 / ncppb 528 / lmg 568 / p 25)
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2026-03-11 Classification: TRANSCRIPTION |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2026-02-18 Classification: TRANSFERASE Ligands: ADP, MG |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2026-02-18 Classification: TRANSFERASE Ligands: ADP, MG |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2026-02-18 Classification: TRANSFERASE Ligands: MG, ADP |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2026-02-18 Classification: TRANSFERASE Ligands: ADP, MG |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2026-01-28 Classification: TRANSFERASE Ligands: ANP |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2026-01-28 Classification: TRANSFERASE Ligands: MG, ANP |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-01-28 Classification: TRANSFERASE |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2026-01-28 Classification: TRANSFERASE Ligands: ATP, MG |
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Structural Basis Of Signal Activation And Transduction By Chitin Elicitor Receptor Kinase 1 In Oryza Sativa
Organism: Oryza sativa japonica group
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2026-01-28 Classification: TRANSFERASE Ligands: ADP, MG |
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Crystal Structure Of Human Glutaminyl Cyclase In Complex With N-(2-(1H-Imidazol-5-Yl)Ethyl)-4-Methoxybenzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: ZN, A1EFY |
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Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With The Inhibitor N-(1H-Benzo[D]Imidazol-5-Yl)-1-Phenylmethanesulfonamide (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2025-03-12 Classification: TRANSFERASE Ligands: ZN, A1D93, GOL, DMS, DMF, PEG |
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Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With The Inhibitor 3-((2-(1H-Imidazol-5-Yl)Ethyl)Carbamoyl)-4-Amino-1,2,5-Oxadiazole 2-Oxide (Compound 13)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2025-03-12 Classification: TRANSFERASE Ligands: ZN, A1D94, DMS, GOL, DMF |
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Crystal Structure Of Human Golgi Resident Glutaminyl Cyclase In Complex With (Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-(Piperidin-4-Yloxy)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.13 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D46 |
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Crystal Structure Of Human Golgi Resident Glutaminyl Cyclase In Complex With (Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-((Tetrahydro-2H-Pyran-4-Yl)Oxy)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.54 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D47 |
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Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With (S)-1-(1H-Benzo[D]Imidazol-5-Yl)-5-(4-Propoxyphenyl)Imidazolidin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.24 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D49 |




















