Search Count: 24
 |
X-Ray Crystal Structure Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A 2-Aryl Benzimidazole Compound And An Internal Aldimine Linked Plp Cofactor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2016-05-04 Classification: TRANSFERASE Ligands: PLP, EL2, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: PLP, EL2, CL, EDO, GOL
 |
X-Ray Crystal Structure At 2.20A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrazolopyrimidinone Fragment And An Internal Aldimine Linked Plp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4VT, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4VT, CL, EDO
 |
X-Ray Crystal Structure At 2.20A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrazolopyrimidinone Fragment And An Internal Aldimine Linked Plp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4VS, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4VS, CL, EDO, GOL
 |
X-Ray Crystal Structure At 2.17A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Triazolopyrimidinone Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4VR, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4VR, EDO
 |
X-Ray Crystal Structure At 1.86A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrazolopyrimidinone Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 775, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 775, CL, EDO, GOL
 |
X-Ray Crystal Structure At 1.82A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Pyrrolidine Amide Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4W6, EDO, CL, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4W6, EDO, CL, GOL, DMS
 |
X-Ray Crystal Structure At 1.70A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A 4-Chloro-2-Fluoro Substituted Pyrazolopyrimidinone Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: PLP, 4W4, EDO, CL, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: PLP, 4W4, EDO, CL, GOL, DMS
 |
N-Terminal Bromodomain Of Human Brd2 With I-Bet726 (Gsk1324726A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: EDO, 73B, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: EDO, 73B, SO4
 |
C-Terminal Bromodomain Of Human Brd2 With I-Bet726 (Gsk1324726A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: 73B, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 73B, SO4
 |
N-Terminal Bromodomain Of Human Brd2 With 1-((2R,4S)-2-Methyl-4-(Phenylamino)-6-(4-(Piperidin-1-Ylmethyl)Phenyl)-3,4-Dihydroquinolin-1(2H)-Yl)Ethanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: 9S3, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 9S3, SO4, DMS
 |
Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2013-10-02 Classification: CELL CYCLE Ligands: H4C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: H4C
 |
Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-10-02 Classification: CELL CYCLE Ligands: L5S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: L5S, EDO
 |
The First Bromodomain Of Human Brd4 In Complex With 3,5 Dimethylisoxaxole Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2013-09-11 Classification: TRANSCRIPTION Ligands: EDO, S5B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: EDO, S5B
 |
The First Bromodomain Of Human Brd4 In Complex With 3,5 Dimethylisoxaxole Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2013-09-11 Classification: TRANSCRIPTION Ligands: EDO, UTH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: EDO, UTH
 |
The First Bromodomain Of Human Brd4 In Complex With 3,5 Dimethylisoxaxole Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-09-11 Classification: TRANSCRIPTION Ligands: EDO, 9BM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: EDO, 9BM
 |
The First Bromodomain Of Human Brd4 In Complex With 3,5 Dimethylisoxaxole Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2013-09-11 Classification: TRANSCRIPTION Ligands: 9B6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: 9B6
 |
N-Terminal Bromodomain Of Human Brd2 With Tbutyl-Phenyl-Amino- Dimethyl-Oxazolyl-Quinoline-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2012-07-04 Classification: PROTEIN BINDING Ligands: EDO, S5B, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: EDO, S5B, SO4, DMS
 |
N-Terminal Bromodomain Of Human Brd2 With Ibet-151
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-07-04 Classification: SIGNALING PROTEIN Ligands: ACT, GOL, 1GH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: ACT, GOL, 1GH
 |
Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gw841819X
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-06-15 Classification: NUCLEAR PROTEIN Ligands: WSH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: WSH, SO4
 |
Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gsk525762 (Ibet)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-06-15 Classification: SIGNALING PROTEIN Ligands: EAM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: EAM, SO4