Search Count: 15
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Crystals Structure Of B-Raf Kinase Domain In Complex With An Imidazopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2017-11-22 Classification: Transferase/Transferase Inhibitor Ligands: 8EN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-22
Ligands: 8EN
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P38 Alpha Mutant C162S In Complex With Cmpd2 [N-(4-Methyl-3-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenyl)-3-(Trifluoromethyl)Benzamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2017-11-15 Classification: TRANSFERASE Ligands: 8EN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: 8EN
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Co-Structure Of Human Glycogen Synthase Kinase Beta With A Selective (5-Imidazol-2-Yl-4-Phenylpyrimidin-2-Yl)[2-(2-Pyridylamino)Ethyl]Amine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-11-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GOL, 65C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-08
Ligands: GOL, 65C
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Discovery Of Imidazo[1,2-A]-Pyridine Inhibitors Of Pan-Pi3 Kinases That Are Efficacious In A Mouse Xenograft Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 5XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: GOL, 5XV
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Structure Of Mcl1 Bound To Brd Inhibitor Ligand 1 At 1.7A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-05-06 Classification: Apoptosis/Inhibitor Ligands: ZN, 865, POP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: ZN, 865, POP
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Structure Of Apo Mbp-Mcl1 At 1.9A
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-05-06 Classification: APOPTOSIS Ligands: MG, EDO, FMT |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: MG, EDO, FMT
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Structure Of Mbp-Mcl1 Bound To Ligand 1 At 2.35A
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-05-06 Classification: APOPTOSIS Ligands: 865, EDO, FMT |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 865, EDO, FMT
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Structure Of Mbp-Mcl1 Bound To Ligand 2 At 1.55A
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2015-05-06 Classification: APOPTOSIS Ligands: 19H, MG, FMT, NA, EDO |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 19H, MG, FMT, NA, EDO
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Structure Of Mbp-Mcl1 Bound To Ligand 4 At 2.4A
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-05-06 Classification: APOPTOSIS Ligands: CL, MG, 3R4 |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: CL, MG, 3R4
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The Structure Of Mbp-Mcl1 Bound To Ligand 5 At 1.9A
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-05-06 Classification: APOPTOSIS Ligands: MG, EDO, FMT, 3R6 |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: MG, EDO, FMT, 3R6
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The Structure Of Mbp-Mcl1 Bound To Ligand 6 At 2.0A
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-05-06 Classification: APOPTOSIS Ligands: 3R7, FMT, MG |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 3R7, FMT, MG
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Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UJ, SO4
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Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UK, SO4
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Co-Crystal Structure Of The Human Kinesin Eg5 With A Novel Tetrahydro-Beta-Carboline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-12-15 Classification: MOTOR PROTEIN Ligands: MG, ADP, L31, NO3, CL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-15
Ligands: MG, ADP, L31, NO3, CL, PEG
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4-(Aminoalkylamino)-3-Benzimidazole-Quinolinones As Potent Chk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2007-03-20 Classification: TRANSFERASE Ligands: SO4, 12C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: SO4, 12C