Search Count: 16
![]() |
Mth1 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: S3O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: S3O
![]() |
Mth1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: 8JF
![]() |
Mth1 In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GN6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: GN6
![]() |
N-Terminal Bromodomain Of Human Brd2 With N-((4-(3-(N-Cyclopentylsulfamoyl)-4-Methylphenyl)-3-Methylisoxazol-5-Yl)Methyl)Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JWA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JWA
![]() |
N-Terminal Bromodomain Of Human Brd2 In Complex With 4,4'-(Quinoline-5,7-Diyl)Bis(3,5-Dimethylisoxazole) Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JWD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JWD, SO4
![]() |
N-Terminal Bromodomain Of Human Brd2 In Complex With N-Cyclopentyl-7-(3,5-Dimethylisoxazol-4-Yl)Quinoline-5-Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JVY
![]() |
C-Terminal Bromodomain Of Human Brd2 In Complex With 4-(2-Cyclopropyl-7-(6-Methylquinolin-5-Yl)-1H-Benzo[D]Imidazol-5-Yl)-3,5-Dimethylisoxazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JW4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JW4, GOL
![]() |
Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2017-11-29 Classification: Transferase/Transferase Inhibitor Ligands: YAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-29
Ligands: YAM
![]() |
Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-12-21 Classification: Transferase/Transferase Inhibitor Ligands: 7FM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: 7FM
![]() |
Crystal Structure Of E. Coli Ccmg
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-03-23 Classification: OXIDOREDUCTASE |
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
![]() |
X-Ray Structure Of The Aquaglyceroporin From Plasmodium Falciparum
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2008-05-27 Classification: MEMBRANE PROTEIN Ligands: BOG, GOL |
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION
Release Date: 2008-05-27
Ligands: BOG, GOL
![]() |
L. Casei Thymidylate Synthase Y261F In Complex With Substrate, Dump
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-03-14 Classification: TRANSFERASE Ligands: UMP |
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION
Release Date: 2006-03-14
Ligands: UMP
![]() |
L. Casei Thymidylate Synthase Y261A In Complex With Substrate, Dump
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-03-14 Classification: TRANSFERASE Ligands: UMP |
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION
Release Date: 2006-03-14
Ligands: UMP
![]() |
Lactobacillus Casei Y261M In Complex With Substrate, Dump
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-03-14 Classification: TRANSFERASE Ligands: UMP |
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION
Release Date: 2006-03-14
Ligands: UMP
![]() |
Lactobacillus Casei Thymidylate Synthase Y261W-Dump Complex
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-03-14 Classification: TRANSFERASE Ligands: UMP |
Organism: Lactobacillus casei
Method: X-RAY DIFFRACTION
Release Date: 2006-03-14
Ligands: UMP
![]() |
Escherichia Coli Y209W Apoprotein
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2006-03-14 Classification: TRANSFERASE Ligands: CO3, PO4, DTT |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2006-03-14
Ligands: CO3, PO4, DTT
