Search Count: 32
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX7, IOD, 1HX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX7, IOD, 1HX
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX9, IOD, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX9, IOD, PEG
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Z237451470
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2023-08-30 Classification: TRANSFERASE Ligands: SAM, WJL, EDO, CL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-30
Ligands: SAM, WJL, EDO, CL, NA
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2023-08-30 Classification: TRANSFERASE Ligands: SAM, WIV, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-30
Ligands: SAM, WIV, CL, EDO
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Allosteric Compound Stl232591
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2023-08-30 Classification: TRANSFERASE Ligands: MTA, ABA, WK5, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-30
Ligands: MTA, ABA, WK5, CL, EDO
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Compound Ideaya Cmpd A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2023-08-30 Classification: TRANSFERASE Ligands: UM6, GOL, MG, SAM, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-30
Ligands: UM6, GOL, MG, SAM, CL
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Human Ido1 In Complex With Compound 4-A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2020-08-26 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: U41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: U41
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Structure Of Human Hdac2 In Complex With Saha (Vorinostat)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-08-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, NA, PG4, SHH, NHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-21
Ligands: ZN, CA, NA, PG4, SHH, NHE
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Structure Of Human Hdac2 In Complex With Inhibitor 4-(Acetylamino)-N-[2-Amino-5-(Thiophen-2-Yl)Phenyl]Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2013-08-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, NA, PG4, 20Y, NHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-21
Ligands: ZN, CA, NA, PG4, 20Y, NHE
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Crystal Structure Of Human Cdk8/Cycc In Complex With Compound 7 (1-[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]Urea)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0SQ, EDO, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0SQ, EDO, FMT
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Crystal Structure Of Human Cdk8/Cycc In Complex With Compound 5 (1-[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]-3-[3-(Morpholin-4-Yl)Propyl]Urea)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0SR, NA, DMS, EDO, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0SR, NA, DMS, EDO, FMT
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Crystal Structure Of Human Cdk8/Cycc In Complex With Compound 1 (N-[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]-4-[2-({[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]Carbamoyl}Amino)Ethyl]Piperazine-1-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0SS, DMS, EDO, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0SS, DMS, EDO, FMT
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Crystal Structure Of Human Cdk8/Cycc In Complex With Compound 4 (1-[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]-3-[2-(Morpholin-4-Yl)Ethyl]Urea)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0ST, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0ST, EDO
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Crystal Structure Of Human Cdk8/Cycc In Complex With Compound 3 (1-[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]-3-(2-Hydroxyethyl)Urea)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0SU, EDO, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0SU, EDO, FMT
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Crystal Structure Of Human Cdk8/Cycc In Complex With Compound 2 (Tert-Butyl [3-({[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]Carbamoyl}Amino)Propyl]Carbamate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0SO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0SO
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Crystal Structure Of Human Cdk8/Cycc In Complex With Compound 11 (1-[3-Tert-Butyl-1-(4-Methylphenyl)-1H-Pyrazol-5-Yl]-3-(5-Hydroxypentyl)Urea)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0SV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0SV, EDO
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Crystal Structure Of Human Cdk8/Cycc In The Dmg-In Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION/INHIBITOR Ligands: 0SW, EDO, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0SW, EDO, FMT
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Crystal Structure Of Human Cdk8/Cycc In The Dmg-In Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-05-01 Classification: TRANSFERASE/TRANSCRIPTION Ligands: FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: FMT
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Endothiapepsin In Complex With A Fragment
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2011-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: F91, GOL, DMS |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: F91, GOL, DMS
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Endothiapepsin In Complex With A Fragment
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2011-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: F90, GOL |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: F90, GOL