Search Count: 36
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Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, NAG, A1JCF, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, NAG, A1JCF, PO4
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Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, NAG, A1JCG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, NAG, A1JCG, PO4
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Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 6 (Oric-533)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, A1JCH, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, A1JCH, PO4
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Crystal Structure Of Egfr Exon20 Insertion Mutant In Complex With Enozertinib (Oric-114)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2025-11-12 Classification: SIGNALING PROTEIN Ligands: A1L8T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1L8T
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Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, VPD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: ZN, CA, VPD
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Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, NAG, VPG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: ZN, CA, NAG, VPG, PO4
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Crystal Structure Of Irak4 In Complex With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: LS7, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: LS7, SO4, GOL
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Structure Of The Irak4 Kinase Domain With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: CA, LRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: CA, LRS
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Structure Of The Irak4 Kinase Domain With Compound 41
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: SO4, LSV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: SO4, LSV
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Structure Of The Irak4 Kinase Domain With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: LTY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: LTY
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Usp7 In Complex With Cpd2 (4-(3-(1-Methylpiperidin-4-Yl)-1,2,4-Oxadiazol-5-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2017-12-13 Classification: HYDROLASE Ligands: AJJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: AJJ, GOL
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Usp7 In Complex With Gne6640 (4-(2-Amino-4-Ethyl-5-(1H-Indazol-5-Yl)Pyridin-3-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JM
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Usp7 In Complex With Gne6776 (6'-Amino-4'-Ethyl-5'-(4-Hydroxyphenyl)-N-Methyl-[3,3'-Bipyridine]-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 8JP
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-09-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 59N
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Crystal Structure Of P21-Activated Kinase 1 (Pak1) In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 6BZ
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound G-5555
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59T
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound Frax1036
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59U, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59U, DMS
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P110Alpha/P85Alpha With Compound 5
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-01-27 Classification: Transferase/Transferase Inhibitor Ligands: 5H2 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H2
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P110Alpha With Gdc-0326
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5, EDO
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P110Delta/P85Alpha With Gdc-0326
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5
