Search Count: 24
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Translation Initiation Factor Eif-2B Complex With The Isohexide Diamine Gsk735
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-03-04 Classification: TRANSLATION Ligands: PRO, SO4, EDO, A1C32 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: PRO, SO4, EDO, A1C32
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Structure Of Crbn:Ikzf2:Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-09-03 Classification: IMMUNE SYSTEM Ligands: A1CBH, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1CBH, ZN
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Structure Of Crbn:Ikzf2:Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2025-09-03 Classification: IMMUNE SYSTEM Ligands: A1CBG, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1CBG, ZN
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Structure Of Ikzf2:Crbn:Compound 5 Ternary Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2025-07-09 Classification: IMMUNE SYSTEM Ligands: A1CAC, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-09
Ligands: A1CAC, ZN
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Structure Of Crbn Tbd Bound To Compound C1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2025-05-28 Classification: IMMUNE SYSTEM Ligands: A1CAV, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1CAV, ZN
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Structure Of Crbn Tbd Bound To Compound C3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2025-05-28 Classification: IMMUNE SYSTEM Ligands: A1CAW, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1CAW, ZN
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Pvtx-405: A Potent, Highly Selective, And Orally Efficacious Molecular Glue Degrader Of Ikzf2 For Cancer Immunotherapy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2025-05-14 Classification: TRANSCRIPTION Ligands: A1A8N, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1A8N, ZN
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1BF5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1BF5, ZN
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1O, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1O, ZN, ACT
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1P, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1P, ZN, ACT
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Rip2 Kinase Catalytic Domain Complex With 2(4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl)Oxy)Ethyl Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: K9T, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: K9T, CA
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Rip2 Kinase Catalytic Domain Complex With 2({4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl}Oxy)Ethan1Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: KA2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: KA2
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Crystal Structure Of Rip1 Kinase In Complex With Gsk3145095
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2019-07-03 Classification: TRANSFERASE Ligands: K8K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-03
Ligands: K8K
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Crystal Structure Of Rip1 Kinase In Complex With A Pyrrolidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2019-05-08 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: M5J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: M5J, SO4
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Crystal Structure Of Rip1 Kinase In Complex With Dhp77
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: JSW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: JSW
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Rip2 Kinase Catalytic Domain Complex With N(4,5Dimethyl1Hpyrazol3Yl)7Methoxy6(2Methylpropane2Sulfonyl)Quinolin4Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-11-07 Classification: TRANSFERASE Ligands: GEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: GEZ
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Rip1 Kinase ( Flag 1-294, C34A, C127A, C233A, C240A) With Gsk772
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-07-05 Classification: transferase/transferase inhibitor Ligands: 7MJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: 7MJ
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The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Compound 3 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GE, SO4
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The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Gsk583 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GD
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Crystal Structure Of Rip1 Kinase With A Benzo[B][1,4]Oxazepin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 65U