Search Count: 44
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Crystal Structure Of Cdk4 Cyclin D1 In Complex With Atirmociclib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2025-03-26 Classification: Transferase/Inhibitor/Cell Cycle Ligands: A1AZ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-26
Ligands: A1AZ4
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Crystal Structure Of Cdk6 In Complex With Atirmociclib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-03-26 Classification: TRANSFERASE Ligands: A1AZ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-26
Ligands: A1AZ4
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Crystal Structure Of Trka (G595R) Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2021-10-13 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
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Crystal Structure Of Trka (G595R) Kinase With Repotrectinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2021-10-13 Classification: TRANSFERASE Ligands: 7GI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: 7GI, SO4
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Crystal Structure Of Trka Kinase With Repotrectinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2021-10-13 Classification: TRANSFERASE Ligands: 7GI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: 7GI, SO4
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Crystal Structure Of Cdk2/Cyclin E In Complex With Pf-06873600
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2021-06-23 Classification: CELL CYCLE Ligands: WG1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-23
Ligands: WG1
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Covalent Complex Of Sars-Cov Main Protease With N-[(2S)-1-({(2S,3S)-3,4-Dihydroxy-1-[(3S)-2-Oxopyrrolidin-3-Yl]Butan-2-Yl}Amino)-4-Methyl-1-Oxopentan-2-Yl]-4-Methoxy-1H-Indole-2-Carboxamide
Organism: Human sars coronavirus
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2020-07-08 Classification: VIRAL PROTEIN Ligands: V2M |
Organism: Human sars coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2020-07-08
Ligands: V2M
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Covalent Complex Of Sars-Cov-2 Main Protease With N-[(2S)-1-({(2S,3S)-3,4-Dihydroxy-1-[(3S)-2-Oxopyrrolidin-3-Yl]Butan-2-Yl}Amino)-4-Methyl-1-Oxopentan-2-Yl]-4-Methoxy-1H-Indole-2-Carboxamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2020-07-08 Classification: VIRAL PROTEIN Ligands: V2M, EDO |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2020-07-08
Ligands: V2M, EDO
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Covalent Complex Of Sars-Cov Main Protease With 4-Methoxy-N-[(2S)-4-Methyl-1-Oxo-1-({(2S)-3-Oxo-1-[(3S)-2-Oxopyrrolidin-3-Yl]Butan-2-Yl}Amino)Pentan-2-Yl]-1H-Indole-2-Carboxamide
Organism: Human sars coronavirus
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2020-07-08 Classification: VIRAL PROTEIN Ligands: V3D, EDO |
Organism: Human sars coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2020-07-08
Ligands: V3D, EDO
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Covalent Complex Of Sars-Cov Main Protease With Ethyl (4R)-4-({N-[(4-Methoxy-1H-Indol-2-Yl)Carbonyl]-L-Leucyl}Amino)-5-[(3S)-2-Oxopyrrolidin-3-Yl]Pentanoate
Organism: Human sars coronavirus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2020-07-08 Classification: VIRAL PROTEIN Ligands: EDO, V34 |
Organism: Human sars coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2020-07-08
Ligands: EDO, V34
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Discovery Of A Novel And Selective Ido-1 Inhibitor Pf-06840003 And Its Characterization As A Potential Clinical Candidate.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2017-12-27 Classification: OXIDOREDUCTASE/Inhibitor Ligands: HEM, AOJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: HEM, AOJ
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Structure Of The Axl Kinase Domain In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2017-07-26 Classification: Transferase/Transferase Inhibitor Ligands: 7YS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: 7YS
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Crystal Structure Of The Mer Kinase Domain In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-07-26 Classification: Transferase/Transferase Inhibitor Ligands: 7YS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: 7YS
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Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-(Propan-2-Yl)-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8BP, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8BP, SO4, GOL
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Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(3-Methoxy-1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-(Propan-2-Yl)-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8AM, SO4, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8AM, SO4, GOL, EDO
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Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With 4-(4-{[2-{[(3S)-1-Acetylpyrrolidin-3-Yl]Amino}-9-(Propan-2-Yl)-9H-Purin-6-Yl]Amino}Phenyl)-1-Methylpiperazin-1-Ium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8BM, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8BM, SO4, GOL
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Crystal Structure Of The Egfr Kinase Domain In Complex With 4-(4-{[2-{[(3S)-1-Acetylpyrrolidin-3-Yl]Amino}-9-(Propan-2-Yl)-9H-Purin-6-Yl]Amino}Phenyl)-1-Methylpiperazin-1-Ium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8BM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8BM
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Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(3-Methoxy-1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-Methyl-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8BS, SO4, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8BS, SO4, GOL, EDO
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The X-Ray Co-Crystal Structure Of Human Cdk6 And Palbociclib.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2016-08-24 Classification: Transferase/Transferase Inhibitor Ligands: LQQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: LQQ
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The X-Ray Co-Crystal Structure Of Human Cdk6 And Abemaciclib.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2016-08-24 Classification: Transferase/Transferase Inhibitor Ligands: 6ZV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: 6ZV