Search Count: 27
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Structure And Function Of The Hypertension Variant A486V Of G Protein-Coupled Receptor Kinase 4 (Grk4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-07-08 Classification: TRANSFERASE Ligands: AN2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-08
Ligands: AN2
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Structure Of Dually Phosphorylated C-Met Receptor Kinase In Complex With An Mk-2461 Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M61 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: M61
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Structure Of The Apo Met Receptor Kinase In The Dually-Phosphorylated, Activated State
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2011-01-19 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
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Structure Of Dually-Phosphorylated Met Receptor Kinase In Complex With An Mk-2461 Analog With Specificity For The Activated Receptor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2011-01-19 Classification: transferase/transferase inhibitor Ligands: Q6W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: Q6W
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Pdk1 In Complex With Inhibitor Mp7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2010-11-24 Classification: TRANSFERASE Ligands: MP7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-24
Ligands: MP7
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Pdk1 In Complex With Inhibitor Mp6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-11-24 Classification: TRANSFERASE Ligands: MP6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-24
Ligands: MP6
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Crystal Structure Of Unphosphorylated P70S6K1 (Form I)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-10-27 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-27
Ligands: STU
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Crystal Structure Of Unphosphorylated P70S6K1 (Form Ii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.43 Å Release Date: 2009-10-27 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-27
Ligands: STU
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Crystal Structure Of Phosphorylated P70S6K1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2009-10-27 Classification: TRANSFERASE Ligands: STU, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-27
Ligands: STU, MN
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Discovery Of Aminoheterocycles As A Novel Beta-Secretase Inhibitor Class
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: B35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: B35
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Crystal Structure Of Chk1 Kinase In Complex With Inhibitor 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-01-20 Classification: TRANSFERASE Ligands: 38M, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: 38M, SO4
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Crystal Structure Of Human Prostasin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2008-10-14 Classification: HYDROLASE Ligands: CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: CL
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Crystal Structure Of Human Prostasin Complexed To 4-Guanidinobenzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-10-14 Classification: HYDROLASE Ligands: GBS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: GBS
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Crystal Structure Of The N-Terminal Kinase Domain Of Human Rsk-1 Bound To Amp-Pcp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-05-13 Classification: TRANSFERASE Ligands: MG, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-05-13
Ligands: MG, ACP
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Crystal Structure Of The N-Terminal Kinase Domain Of Human Rsk1 Bound To Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-05-13 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-05-13
Ligands: STU
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Crystal Structure Of The N-Terminal Kinase Domain Of Human Rsk1 Bound To Purvalnol A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-05-13 Classification: TRANSFERASE Ligands: P01 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-05-13
Ligands: P01
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Crystal Structure Of Human Beta Secretase Complexed With I21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-04-29 Classification: HYDROLASE Ligands: I21 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-29
Ligands: I21
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Crystal Structure Of Human Beta Secretase Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-04-22 Classification: HYDROLASE Ligands: SO4, 35A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: SO4, 35A
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Crystal Structure Of Chek1 In Complex With Inhibitor 2A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-03-18 Classification: TRANSFERASE Ligands: 7CS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-18
Ligands: 7CS
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Crystal Structure Of Chek1 In Complex With Inhibitor 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-03-18 Classification: TRANSFERASE Ligands: 582 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-18
Ligands: 582
