Search Count: 26
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Crystal Structure Of The Complex Between Vhl, Elonginb, Elonginc, And Compound 5
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2024-05-29 Classification: TRANSCRIPTION Ligands: TFA, PEG, EDO, ACT, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: TFA, PEG, EDO, ACT, DMS
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Crystal Structure Of The Complex Between Vhl, Elonginb, Elonginc, And Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2024-05-29 Classification: TRANSCRIPTION Ligands: EDO, DMS, CL, A1ARP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, DMS, CL, A1ARP
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Crystal Structure Of Human Mcl-1 In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-02-14 Classification: TRANSFERASE Ligands: WXW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: WXW
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Co-Crystal Structure Of Perk With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2022-11-30 Classification: TRANSFERASE/Inhibitor Ligands: WPB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: WPB
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Co-Crystal Structure Of Perk With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2022-11-30 Classification: TRANSFERASE Ligands: WPX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: WPX
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Co-Crystal Structure Of Perk With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2022-11-30 Classification: TRANSFERASE Ligands: WQ2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: WQ2
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Kras G12C In Complex With G-2897
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-03-16 Classification: HYDROLASE/Immune System Ligands: Z07, GDP, MG, ACT, CAD, P15, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: Z07, GDP, MG, ACT, CAD, P15, EDO, DMS
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Crystal Structure Of Kas G12C In Complex With 2H11 Clamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-03-16 Classification: Hydrolase/Immune System Ligands: GDP, MG, CAC, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: GDP, MG, CAC, EDO
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Crystal Structure Of Gne-1952 Alkylated Kras G12C In Complex With 2H11 Clamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-03-16 Classification: Hydrolase/Immune System Ligands: MKZ, GDP, MG, GOL, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: MKZ, GDP, MG, GOL, EDO, SO4
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Crystal Structure Of Kras G12C In Complex With Gne-1952
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-03-16 Classification: HYDROLASE Ligands: MKZ, GDP, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: MKZ, GDP, MG, GOL
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Lc3A In Complex With Fragment 1-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2022-01-12 Classification: HYDROLASE Ligands: JO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: JO4, GOL
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Lc3A In Complex With Fragment 2-3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2022-01-12 Classification: HYDROLASE Ligands: 2LZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: 2LZ
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Lc3A In Complex With Fragment 2-10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2022-01-12 Classification: HYDROLASE Ligands: 2JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: 2JI
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Co-Crystal Structure Of Perk With Inhibitor (R)-2-Amino-N-Cyclopropyl-5-(4-(2-(3,5-Difluorophenyl)-2-Hydroxyacetamido)-2-Methylphenyl)Nicotinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: Z6P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: Z6P
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Structure Of Tak1 In Complex With Compound 54
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-04-07 Classification: TRANSFERASE Ligands: GOL, DMS, URW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: GOL, DMS, URW
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Structure Of Tak1 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-04-07 Classification: TRANSFERASE Ligands: GOL, DMS, UWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: GOL, DMS, UWZ
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Ternary Complex Of Vhl/Brd4-Bd1/Compound9 (4-(3,5-Difluoropyridin-2-Yl)-N-(11-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-Methylthiazol-5-Yl)Benzyl)Carbamoyl)Pyrrolidin-1-Yl)-3,3-Dimethyl-1-Oxobutan-2-Yl)Amino)-11-Oxoundecyl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-02-24 Classification: PEPTIDE BINDING PROTEIN Ligands: WEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEP
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Brd4-Bd1 Compound6 (Methyl 4-(3,5-Difluoropyridin-2-Yl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2021-02-24 Classification: CELL CYCLE Ligands: WEM, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEM, GOL
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A New Autotaxin Inhibitor For The Treatment Of Idiopathic Pulmonary Fibrosis: A Clinical Candidate Discovered Using Dna-Encoded Chemistry
Organism: Pan troglodytes
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2020-07-08 Classification: LIPID BINDING PROTEIN Ligands: NAG, SKV, ZN, CA, MG, SCN, CL, IOD |
Organism: Pan troglodytes
Method: X-RAY DIFFRACTION
Release Date: 2020-07-08
Ligands: NAG, SKV, ZN, CA, MG, SCN, CL, IOD
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C-Met In Complex With Osi Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-04-30 Classification: TRANSFERASE Ligands: 1RU, GBL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-30
Ligands: 1RU, GBL