Search Count: 15
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Crystal Structure Of Tankyrase 1 With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2C6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: ZN, 2C6
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Co-Crystal Structure Of Tankyrase 1 With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2C8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: ZN, 2C8
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Co-Crystal Structure Of Tankyrase 1 With Compound 49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 2D6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: ZN, 2D6
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Co-Crystal Structure Of Tnks1 With Compound 52 [N~2-(5-Chloro-2-Methoxyphenyl)-N-[Trans-4-(2-Oxo-2,3-Dihydro-1H-Benzimidazol-1-Yl)Cyclohexyl]Glycinamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-06-05 Classification: Transferase/Transferase Inhibitor Ligands: ZN, K4E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: ZN, K4E
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Co-Crystal Structure Of Tnks1 With Compound 18 [4-[(4S)-5,5-Dimethyl-2-Oxo-4-Phenyl-1,3-Oxazolidin-3-Yl]-N-(Quinolin-8-Yl)Benzamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-06-05 Classification: Transferase/Transferase Inhibitor Ligands: ZN, K4F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: ZN, K4F
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Crystal Structure Of Pi3K-Gamma In Complex With Imidazopyridazine 19E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2013-04-10 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 0U0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: SO4, 0U0
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Crystal Structure Of Human Pi3K-Gamma In Complex With Amg511
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-08-29 Classification: Transferase/Inhibitor Ligands: SO4, 14K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: SO4, 14K
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Crystal Structure Of Human Pi3K-Gamma In Complex With A Pyridyl-Triazine-Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2012-08-08 Classification: Transferase/Inhibitor Ligands: SO4, F1S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: SO4, F1S
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Crystal Structure Of Pi3K-Gamma In Complex With Imidazopyridine 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-07-18 Classification: Transferase/Inhibitor Ligands: SO4, 0TZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-18
Ligands: SO4, 0TZ
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Crystal Structure Of Human Pi3K-Gamma In Complex With A Pyridyl-Triazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2012-05-16 Classification: Transferase/Inhibitor Ligands: SO4, 0KO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: SO4, 0KO
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Crystal Structure Of Pi3K-Gamma In Complex With A Quinoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2011-06-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 2NQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-08
Ligands: SO4, 2NQ
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Crystal Structure Of Pi3K-Gamma In Complex With Triazine-Benzimidazole 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, QAQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SO4, QAQ
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Crystal Structure Of Pi3K-Gamma In Complex With Triazine-Benzimidazole 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, QAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SO4, QAR
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Crystal Structure Of Pi3K-Gamma In Complex With Benzothiazole 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QJZ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: QJZ, SO4
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Crystal Structure Of Pi3K-Gamma In Complex With Benzothiazole 82
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, QK0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SO4, QK0
