Search Count: 39
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Fragments Bound To Hiv-1 Integrase
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, SO4, 0NX |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, SO4, 0NX
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Hiv-1 In Core Domain In Complex With N-Methyl-1-(4-Methyl-2-Phenyl-1,3-Thiazol-5-Yl)Methanamine
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, CL, SO4, MMJ |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, CL, SO4, MMJ
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Hiv-1 In Core Domain In Complex With (1-Methyl-5-Phenyl-1H-Pyrazol-4-Yl)Methanol
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, BCK, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, BCK, SO4
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Hiv-1 In Core Domain In Complex With 4-(1H-Pyrrol-1-Yl)Aniline
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, SO4, SNU |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, SO4, SNU
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Hiv-1 In Core Domain In Complex With (3R)-3,4-Dihydro-2H-Chromen-3-Ylmethanol
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, CL, SO4, BCU |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, CL, SO4, BCU
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Hiv-1 In Core Domain In Complex With 6-Fluoro-1,3-Benzothiazol-2-Amine
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FBB |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: FBB
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Hiv-1 In Core Domain In Complex With 1-Benzothiophen-6-Amine 1,1-Dioxide
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, SO4, MWP |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, SO4, MWP
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Hiv-1 In Core Domain In Complex With 6-Fluoro-4H-1,3-Benzodioxine-8-Carboxylic Acid
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, SO4, FBG |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, SO4, FBG
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Hiv-1 In Core Domain In Complex With (5-Methyl-3-Phenyl-1,2-Oxazol-4-Yl)Methanol
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, SO4, MPK |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, SO4, MPK
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Hiv-1 In Core Domain In Complex With 5-Methyl-3-Phenyl-1,2-Oxazole-4-Carboxylic Acid
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, SO4, MOK |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, SO4, MOK
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Hiv-1 In Core Domain In Complex With [1-(4-Fluorophenyl)-5-Methyl-1H-Pyrazol-4-Yl]Methanol
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, CL, SO4, FMQ |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, CL, SO4, FMQ
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Hiv-1 In Core Domain In Complex With 2,3-Dihydro-1,4-Benzodioxin-5-Ylmethanol
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, CL, SO4, DBJ |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, CL, SO4, DBJ
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Hiv-1 Integrase Core Domain In Complex With 2,1,3-Benzothiadiazol-4-Amine
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-01-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD, SO4, BTE |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CD, SO4, BTE
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Parallel Screening Of A Low Molecular Weight Compound Library: Do Differences In Methodology Affect Hit Identification
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: 0MB, SO4, EDO, CL, GOL, TAM |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: 0MB, SO4, EDO, CL, GOL, TAM
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Parallel Screening Of A Low Molecular Weight Compound Library: Do Differences In Methodology Affect Hit Identification
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: SO4, ACY, GOL, I2E |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: SO4, ACY, GOL, I2E
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Parallel Screening Of A Low Molecular Weight Compound Library: Do Differences In Methodology Affect Hit Identification
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: SO4, ACT, EDO, GOL, AKH |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: SO4, ACT, EDO, GOL, AKH
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Parallel Screening Of A Low Molecular Weight Compound Library: Do Differences In Methodology Affect Hit Identification
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: SO4, EDO, TAM, Q6T, ACY |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: SO4, EDO, TAM, Q6T, ACY
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Parallel Screening Of A Low Molecular Weight Compound Library: Do Differences In Methodology Affect Hit Identification
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: SO4, CL, GOL, ICO, ACY, EDO |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: SO4, CL, GOL, ICO, ACY, EDO
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Parallel Screening Of A Low Molecular Weight Compound Library: Do Differences In Methodology Affect Hit Identification
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: SO4, ACY, EDO, TAM, Z5P |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: SO4, ACY, EDO, TAM, Z5P
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Small Molecule Inhibitors Of The Ledgf Site Of Hiv Integrase Identified By Fragment Screening And Structure Based Design.
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-12-05 Classification: TRANSFERASE Ligands: SO4, GOL, PX3, ACT |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-12-05
Ligands: SO4, GOL, PX3, ACT
