Search Count: 14
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: 9JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: 9JI
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (43)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVO
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (44)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVS
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVR
![]() |
Kit Kinase Domain In Complex With A Pyrrolotriazine-Based Compound (11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVQ
![]() |
Kit Kinase Domain In Complex With An Aminopyrimidine-Based Compound (15)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JV1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JV1
![]() |
Kit Kinase Domain In Complex With A Pyrrolopyrimidine-Based Compound (17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVP
![]() |
Kit Kinase Domain In Complex With A 6-,7-Dimethoxyquinoline-Based Compound (19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVT
![]() |
Kit Kinase Domain In Complex With A 7-Methylquinazoline-Based Compound (25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVW
![]() |
Kit Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (33)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVV
![]() |
Kit Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (34)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVZ
![]() |
Kit Kinase Domain In Complex With A Quinoline-3-Carbonitrile-Based Compound (38)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVY
![]() |
Kit Kinase Domain In Complex With A Methyl Quinazoline-7-Carboxylate-Based Compound (41)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JV0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JV0
![]() |
Kit Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVR
